Adrenergic α1 Receptor Antagonists
| Cat. No. | Product Name / Activity |
|---|---|
| 5940 | AdTx1 |
| Selective, high affinity, non-competitive α1A adrenoceptor antagonist | |
| 3305 | Alfuzosin hydrochloride |
| Uroselective α1 antagonist | |
| 1006 | BMY 7378 dihydrochloride |
| Selective α1D antagonist | |
| 2685 | Carvedilol |
| Potent α1 antagonist; also potent and non-selective β antagonist | |
| 2964 | Doxazosin mesylate |
| α1 antagonist | |
| 0535 | HEAT hydrochloride |
| Highly selective α1 antagonist | |
| 0545 | Ifenprodil hemitartrate |
| α1 antagonist. Also NMDA antagonist and σ ligand | |
| 0661 | 2-MPMDQ |
| Potent, selective α1 antagonist. Also σ2 ligand | |
| 0597 | Naftopidil hydrochloride |
| α1 antagonist | |
| 1124 | (R)-(-)-Niguldipine hydrochloride |
| α1 antagonist, L-type Ca2+ channel blocker. Less active enantiomer of Niguldipine hydrochloride (Cat. No. 1123) | |
| 1123 | (S)-(+)-Niguldipine hydrochloride |
| α1 antagonist, L-type Ca2+ channel blocker | |
| 0627 | 2-PMDQ |
| Potent, selective α1 antagonist | |
| 0623 | Prazosin hydrochloride |
| α1 and α2B antagonist; also MT3 antagonist | |
| 3284 | Rec 15/2615 dihydrochloride |
| Selective α1B antagonist | |
| 1325 | RS 100329 hydrochloride |
| Potent, subtype-selective α1A antagonist | |
| 0985 | RS 17053 hydrochloride |
| α1A antagonist | |
| 6663 | Silodosin |
| Selective α1A antagonist | |
| 2398 | SNAP 5089 |
| Subtype-selective α1A antagonist | |
| 3050 | Tamsulosin hydrochloride |
| Selective α1A antagonist | |
| 1506 | Terazosin hydrochloride |
| α1 and α2B antagonist (α1 > α2B). Orally active | |
| 6336 | Trazodone hydrochloride |
| 5-HT2A and α1 adrenoceptor antagonist; also enhances neural differentiation; antidepressant and neuroprotectant | |
| 1772 | Urapidil hydrochloride |
| α1 antagonist; also 5-HT1A receptor agonist | |
| 0946 | WB 4101 hydrochloride |
| α1A antagonist |
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