The adrenergic β2 receptor (β2-adrenoceptor) is a member of the adrenergic receptor group of G-protein-coupled receptors that also includes α1A, α1B, α1D, α2A, α2B, α2C, β1 and β3. They are located primarily in the CNS, heart, kidney and muscle.
Agonists |
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Cat No | Product Name / Activity |
6219 | Arformoterol tartrate |
Long-acting β2 agonist (LABA) | |
1448 | Formoterol hemifumarate |
Potent and selective β2 agonist | |
1102 | Procaterol hydrochloride |
Potent β2 agonist | |
0634 | Salbutamol hemisulfate |
β agonist (β2 > β1) | |
4712 | Salmeterol xinafoate |
Long-acting β2 agonist; bronchodilator | |
1051 | Zinterol hydrochloride |
Selective β2 agonist | |
Inverse Agonists |
|
Cat No | Product Name / Activity |
0821 | ICI 118,551 hydrochloride |
Very selective β2 inverse agonist | |
Ligand Sets |
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Cat No | Product Name / Activity |
1873 | β-Adrenoceptor Agonist Tocriset™ |
Selection of 3 β-adrenoceptor agonists (Cat. Nos. 0948, 1747 and 1660) | |
1874 | β-Adrenoceptor Antagonist Tocriset™ |
Selection of 3 β-adrenoceptor antagonists (Cat. Nos. 1024, 0821 and 1511) |
The adrenergic β2 receptor (β2-adrenoceptor) is a member of the adrenergic receptor group of G-protein-coupled receptors that also includes α1A, α1B, α1D, α2A, α2B, α2C, β1 and β3. They are located primarily in the CNS, heart, kidney and muscle where they are involved in smooth muscle relaxation (e.g. bronchodilation). The human adrenergic β2 receptor gene has been localized to chromosome 5 (5q31-q32)
Tocris offers the following scientific literature for Adrenergic β2 Receptors to showcase our products. We invite you to request* or download your copy today!
*Please note that Tocris will only send literature to established scientific business / institute addresses.
Major depressive disorder is characterized by depressed mood and a loss of interest and/or pleasure. Updated in 2015 this poster highlights presynaptic and postsynaptic targets for the potential treatment of major depressive disorder, as well as outlining the pharmacology of currently approved antidepressant drugs.