Bromodomain Inhibitors

Cat. No. Product Name / Activity
7757 AZ 13824374
Potent and selective ATAD2 bromodomain inhibitor
5970 BAY 299
Potent and selective BRD1 and TAF1 inhibitor
5266 BAZ2-ICR
Selective BAZ2 inhibitor
5590 BI 9564
Potent and selective BRD9 and BRD7 inhibitor; orally active
4758 Bromosporine
Broad spectrum bromodomain inhibitor
7139 CeMMEC1
TAF1 inhibitor
5331 CPI 203
BET bromodomain inhibitor; arrests cell cycle at G1 phase
7644 FHT 1015
Potent and selective SMARCA4/2 inhibitor
7645 FHT 2344
Potent SMARCA2/4 inhibitor
6198 GSK 6853
Potent and selective BRPF1 inhibitor
4650 I-BET 151 dihydrochloride
BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes
6521 I-BET 762
Potent and high affinity BET bromodomain inhibitor; anti-inflammatory; orally bioavailable.
5591 I-BRD9
Potent and selective BRD9 inhibitor
7458 iBET-BD2
Potent and selective pan-BD2 inhibitor; orally bioavailable
4695 Ischemin sodium salt
CBP inhibitor; cell permeable
4499 (+)-JQ1
Potent and selective BET bromodomain inhibitor; cell permeable
6251 L Moses dihydrochloride
High affinity and selective PCAF bromodomain inhibitor
6068 Lin28 1632
Bromodomain inhibitor; also RNA binding protein Lin28 inhibitor and promotes mESC differentiation
5496 LP 99
Selective BRD7 and BRD9 inhibitor
5173 MS 436
Potent and selective BRD4(1) inhibitor
5546 NI 57
Potent and selective BRPF bromodomain inhibitor
7482 NVS MLLT-1
Selective MLLT1/3 inhibitor
5744 NVS-CECR2-1
Potent and selective CECR2 inhibitor
5289 OF 1
Selective BRPF1B and BRPF2 inhibitor
6181 OTX 015
BET bromodomain inhibitor; orally bioavailable
4928 OXF BD 02
Selective BRD4(1) inhibitor
4445 PFI 1
BET bromodomain inhibitor
5072 PFI 3
Potent and selective SMARCA2/4 and polybromo 1 inhibitor
Potent and selective SMARCA2/4 and PB1(bromo 5)-selective SWI/SNF bromodomain inhibitor
4889 SGC-CBP30
Potent CBP/p300 BRD inhibitor
6670 TP 238
CECR2 and BPTF/FALZ inhibitor
6000 TP 472
Potent BRD9/7 inhibitor
4132 XMD 8-92
BRD4 inhibitor; also ERK5/BMK1 inhibitor