Bromodomain Inhibitors
| Cat. No. | Product Name / Activity |
|---|---|
| 7757 | AZ 13824374 |
| Potent and selective ATAD2 bromodomain inhibitor | |
| 5970 | BAY 299 |
| Potent and selective BRD1 and TAF1 inhibitor | |
| 5266 | BAZ2-ICR |
| Selective BAZ2 inhibitor | |
| 5590 | BI 9564 |
| Potent and selective BRD9 and BRD7 inhibitor; orally active | |
| 4758 | Bromosporine |
| Broad spectrum bromodomain inhibitor | |
| 8892 | CCS 1477 |
| Selective p300/CBP bromodomain inhibitor | |
| 7139 | CeMMEC1 |
| TAF1 inhibitor | |
| 5331 | CPI 203 |
| BET bromodomain inhibitor; arrests cell cycle at G1 phase | |
| 7644 | FHT 1015 |
| Potent and selective SMARCA4/2 inhibitor | |
| 7645 | FHT 2344 |
| Potent SMARCA2/4 inhibitor | |
| 6198 | GSK 6853 |
| Potent and selective BRPF1 inhibitor | |
| 4650 | I-BET 151 dihydrochloride |
| BET bromodomain inhibitor; also promotes differentiation of hiPSCs into megakaryocytes | |
| 6521 | I-BET 762 |
| Potent and high affinity BET bromodomain inhibitor; anti-inflammatory; orally bioavailable. | |
| 5591 | I-BRD9 |
| Potent and selective BRD9 inhibitor | |
| 7458 | iBET-BD2 |
| Potent and selective pan-BD2 inhibitor; orally bioavailable | |
| 4499 | (+)-JQ1 |
| Potent and selective BET bromodomain inhibitor; cell permeable | |
| 6251 | L Moses dihydrochloride |
| High affinity and selective PCAF bromodomain inhibitor | |
| 5496 | LP 99 |
| Selective BRD7 and BRD9 inhibitor | |
| 5546 | NI 57 |
| Potent and selective BRPF bromodomain inhibitor | |
| 7482 | NVS MLLT-1 |
| Selective MLLT1/3 inhibitor | |
| 5744 | NVS-CECR2-1 |
| Potent and selective CECR2 inhibitor | |
| 6181 | OTX 015 |
| BET bromodomain inhibitor; orally bioavailable | |
| 4445 | PFI 1 |
| BET bromodomain inhibitor | |
| 5072 | PFI 3 |
| Potent and selective SMARCA2/4 and polybromo 1 inhibitor | |
| 7460 | SGC SMARCA-BRDVIII |
| Potent and selective SMARCA2/4 and PB1(bromo 5)-selective SWI/SNF bromodomain inhibitor | |
| 4889 | SGC-CBP30 |
| Potent CBP/p300 BRD inhibitor | |
| 6670 | TP 238 |
| CECR2 and BPTF/FALZ inhibitor | |
| 6000 | TP 472 |
| Potent BRD9/7 inhibitor | |
| 4132 | XMD 8-92 |
| BRD4 inhibitor; also ERK5/BMK1 inhibitor |
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