PI 3-kinase Inhibitors

Cat No Product Name / Activity
5595 A66
Potent and selective PI 3-kinase p110α inhibitor
3671 AS 252424
Selective inhibitor of PI 3-kinase γ
3578 AS 605240
Potent and selective PI 3-kinase γ (PI 3-Kγ) inhibitor
4839 AZD 6482
Potent and selective PI 3-Kβ inhibitor
3606 BAG 956
Dual PI 3-kinase and PDPK1 (PDK1) inhibitor
4674 CZC 24832
Selective inhibitor of PI 3-kinase γ
4702 ETP 45658
Potent PI 3-kinase inhibitor; also inhibits DNA-PK and mTOR
4026 GSK 1059615
Potent PI 3-kinase inhibitor
4840 KU 0060648
Dual DNA-PK and PI 3-K inhibitor
5835 LTURM 36
PI 3-kinase δ inhibitor
1130 LY 294002 hydrochloride
Prototypical PI 3-kinase inhibitor; also inhibits other kinases
2418 LY 303511
Negative control of LY 294002 (Cat. No. 1130)
3977 3-Methyladenine
Class III PI 3-kinase inhibitor; also inhibits autophagy
4820 PF 04691502
Potent and selective dual PI 3-K/mTOR inhibitor
4823 PF 05212384
Potent and selective dual PI 3-K/mTOR inhibitor
2930 PI 103 hydrochloride
Inhibitor of PI 3-kinase, mTOR and DNA-PK
5919 PI 3065
Potent and selective PI 3-kinase p110δ inhibitor
2814 PI 828
PI 3-kinase inhibitor, more potent than LY 294002 (Cat. No. 1130)
6440 PIK 93
Potent PI 3-Kγ, PI 3-Kα and PI 4-KIIIβ inhibitor
3894 PP 121
Dual kinase inhibitor; inhibits PI 3-K family kinases
1125 Quercetin
Non-selective PI 3-kinase inhibitor
6036 STK16-IN-1
PI 3Kδ and PI 3Kγ kinase inhibitor; also inhibits mTOR and STK16 kinases
6079 TC KHNS 11
Potent and selective PI 3-kinase δ inhibitor; orally bioavailable
4264 TG 100713
PI 3-kinase inhibitor
5832 TGX 221
Potent and selective PI 3-kinase β inhibitor
1232 Wortmannin
Potent, irreversible inhibitor of PI 3-kinase. Also inhibitor of PLK1