| Cat. No. |
Product Name / Activity |
| 6167 |
A 196 |
| Potent and selective SUV420H1/H2 inhibitor |
| 7648 |
AS 99 New |
| Selective ASH1L histone methyltransferase inhibitor |
| 5991 |
BAY 598 |
| Potent and selective SMYD2 inhibitor |
| 6561 |
BAY 6035 |
| Potent and selective SMYD3 inhibitor |
| 6665 |
BI 9321 |
| Nuclear receptor-binding SET domain (NSD) 3 antagonist; selectively binds PWWP1 domain |
| 4504 |
Chaetocin |
| SUV39H1 inhibitor |
| 7762 |
EED 226 |
| Potent and selective EED inhibitor |
| 5567 |
EPZ 004777 |
| Highly potent DOT1L inhibitor |
| 5648 |
Hydroxychloroquine sulfate |
| PRC2 inhibitor; also autophagy inhibitor and TLR9 inhibitor |
| 6803 |
MRK 740 |
| Potent PRDM9 inhibitor |
| 4892 |
(R)-PFI 2 hydrochloride |
| Potent and selective SETD7 inhibitor |
| 5400 |
(S)-PFI 2 hydrochloride |
| Negative control of (R)-PFI 2 hydrochloride (Cat. No. 4892) |
| 2609 |
Ryuvidine |
| SETD8 inhibitor; also CDK4 inhibitor |
| 4541 |
SGC 0946 |
| Highly potent and selective DOT1L inhibitor; cell permeable |