Other Lysine Methyltransferases

Products
Background
Literature

Antagonists

Cat. No. Product Name / Activity
6665 BI 9321
Nuclear receptor-binding SET domain (NSD) 3 antagonist; selectively binds PWWP1 domain

Inhibitors

Cat. No. Product Name / Activity
6167 A 196
Potent and selective SUV420H1/H2 inhibitor
5991 BAY 598
Potent and selective SMYD2 inhibitor
6561 BAY 6035
Potent and selective SMYD3 inhibitor
4504 Chaetocin
SUV39H1 inhibitor
0996 Cyproheptadine hydrochloride
SETD7/9 inhibitor; also 5HT2 antagonist
5567 EPZ 004777
Highly potent DOT1L inhibitor
5365 LLY 507
Potent SMYD2 inhibitor
4892 (R)-PFI 2 hydrochloride
Potent and selective SETD7 inhibitor
5400 (S)-PFI 2 hydrochloride
Negative control of (R)-PFI 2 hydrochloride (Cat. No. 4892)
2609 Ryuvidine
SETD8 inhibitor; also CDK4 inhibitor
4541 SGC 0946
Highly potent and selective DOT1L inhibitor; cell permeable

Other

Cat. No. Product Name / Activity
4707 MI 2 dihydrochloride
Menin-MLL interaction inhibitor
6096 UNC 3866
High affinity CBX4 and CBX7 inhibitor

External sources of pharmacological information for Other Lysine Methyltransferases :

    Literature for Other Lysine Methyltransferases

    Tocris offers the following scientific literature for Other Lysine Methyltransferases to showcase our products. We invite you to request* or download your copy today!

    *Please note that Tocris will only send literature to established scientific business / institute addresses.


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