Glutamate Transporter Inhibitors

Cat. No. Product Name / Activity
0271 cis-ACBD
Potent, selective L-glutamate uptake inhibitor
0332 L-CCG-lll
Potent, competitive glutamate uptake inhibitor
0846 Chicago Sky Blue 6B
Potent inhibitor of L-glutamate uptake into synaptic vesicles; also inhibits MIF
3697 7-Chlorokynurenic acid sodium salt
Potent competitive inhibitor of L-glutamate uptake. Sodium salt of 7-Chlorokynurenic acid (Cat. No. 0237)
0237 7-Chlorokynurenic acid
Potent competitive inhibitor of L-glutamate uptake
0111 Dihydrokainic acid
EAAT2 (GLT-1)-selective non-transportable inhibitor of L-glutamate and L-aspartate uptake
0845 Evans Blue tetrasodium salt
Potent inhibitor of L-glutamate uptake into synaptic vesicles; also non-NMDA iGluR antagonist; P2X antagonist
2217 (±)-HIP-A
Potent, non-competitive EAAT inhibitor
2218 (±)-HIP-B
Potent, non-competitive EAAT inhibitor
0183 L-(-)-threo-3-Hydroxyaspartic acid
Transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor
0811 (±)-threo-3-Methylglutamic acid
EAAT2 and EAAT4 blocker
0973 MPDC
Potent inhibitor of L-glutamate uptake. Less activity as a substrate compared to its parent compound, L-trans-2,4-PDC (Cat. No. 0298)
0298 L-trans-2,4-PDC
Transportable EAAT1-4 inhibitor/non-transportable EAAT5 inhibitor
0903 SYM 2081
Inhibits EAAT2. Also kainate receptor agonist
1223 DL-TBOA
Selective non-transportable inhibitor of EAATs
2532 TFB-TBOA
High affinity EAAT1 and EAAT2 blocker
3490 UCPH 101
Selective non-substrate EAAT1 inhibitor
2652 WAY 213613
Potent, non-substrate EAAT2 inhibitor