CaV1.x Channel (L-type) Blockers

Cat. No. Product Name / Activity
2571 Amlodipine besylate
CaV1.x blocker
1545 (R)-(+)-Bay K 8644
CaV1.x blocker; (R)-(+)-enantiomer of (±)-Bay K 8644
2629 Cilnidipine
Dual CaV1.x and CaV2.x blocker
6170 Cinacalcet hydrochloride
CaV1.x blocker; also CaSR allosteric agonist and CYP2D2 inhibitor
0685 Diltiazem hydrochloride
CaV1.x blocker
3733 Efonidipine hydrochloride monoethanolate
CaV1.x and CaV3.x blocker
2960 Felodipine
CaV1.x blocker
6407 Fendiline Hydrochloride
CaV1.x blocker; also K-Ras inhibitor
2004 Isradipine
CaV1.x blocker
2959 Lercanidipine hydrochloride
CaV1.x blocker
0840 Loperamide hydrochloride
CaV1.x and CaV2.x blocker; also peripherally acting μ agonist
1075 Nifedipine
CaV1.x blocker
1124 (R)-(-)-Niguldipine hydrochloride
CaV1.x blocker; also α1A antagonist; less active enantiomer of (S)-(+)-Niguldipine
1123 (S)-(+)-Niguldipine hydrochloride
CaV1.x blocker; also α1A antagonist
5711 Nilvadipine
CaV1.x blocker; also Syk kinase inhibitor
0600 Nimodipine
CaV1.x blocker
0601 Nitrendipine
CaV1.x blocker
1806 SR 33805 oxalate
CaV1.x blocker; binds allosterically to distinct site
0654 Verapamil hydrochloride
CaV1.x blocker