Phosphodiesterase Inhibitors
| Cat. No. | 产品名称/活性 |
|---|---|
| 6313 | A 33 |
| Potent and selective PDE4B inhibitor | |
| 2237 | BRL 50481 |
| Selective PDE7 inhibitor | |
| 2793 | Caffeine |
| Cyclic nucleotide PDE inhibitor | |
| 0915 | Cilostamide |
| PDE3 inhibitor | |
| 0691 | Dipyridamole |
| PDE5/6/8/10/11 inhibitor | |
| 1261 | EHNA hydrochloride |
| PDE2 inhibitor | |
| 1693 | Enoximone |
| PDE3 inhibitor | |
| 5202 | Furamidine dihydrochloride |
| TDP-1 inhibitor; PRMT1 inhibitor | |
| 4165 | Gisadenafil besylate |
| Potent PDE5 inhibitor; orally bioavailable | |
| 2845 | IBMX |
| PDE inhibitor (non-selective) | |
| 1694 | Ibudilast |
| PDE inhibitor (non-selective) | |
| 3053 | Mesopram |
| Orally active PDE4 inhibitor | |
| 5915 | PF 04449613 |
| Potent PDE9 inhibitor; brain penetrant | |
| 6024 | PF 04671536 hydrochloride |
| Potent and selective PDE8B/8A inhibitor | |
| 6405 | PF 05180999 |
| Potent and selective PDE2A inhibitor | |
| 4525 | Piclamilast |
| Potent and selective PDE4 inhibitor | |
| 0415 | Ro 20-1724 |
| PDE4 inhibitor | |
| 0905 | Rolipram |
| PDE4 inhibitor | |
| 1349 | (R)-(-)-Rolipram |
| PDE4 inhibitor. More active enantiomer of rolipram (Cat. No. 0905) | |
| 3784 | Sildenafil citrate |
| Potent PDE5 inhibitor; orally active | |
| 6311 | Tadalafil |
| Potent and highly selective PDE5 inhibitor; orally bioavailable | |
| 2337 | Trequinsin hydrochloride |
| Highly potent PDE3 inhibitor | |
| 0947 | Zaprinast |
| PDE5/6/9/11 inhibitor |