New Products

View all new products by date added

Search for new products by date added, alphabetically, or by pharmacological action.

New products are an essential component of our range. Introductions are made on an ongoing basis, with hundreds of new small molecules and peptides being added every year. Our aim is to find the latest, otherwise unobtainable research tools, and bring them to the market as quickly as we can. New products can be identified throughout the Tocris website by the symbol.

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Cat. No. 产品名称/活性 Date Added
7105 VH 032 amide-PEG5-acid Nov 2020
VHL ligand with PEG linker and terminal acid for onward chemistry
7258 Gefitinib-based PROTAC® 3 Nov 2020
Potent EGFR Degrader
7303 iHAP1 Nov 2020
Allosteric activator of protein phosphatase 2A (PP2A)
7255 ARCC 4 negative control Nov 2020
Negative control for ARCC 4 (Cat. No. 7254)
7197 JHU 37152 Nov 2020
High affinity and highly potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant
7254 ARCC 4 Nov 2020
Potent and selective androgen receptor degrader
7213 Pomalidomide 4'-PEG4-acid Nov 2020
Cereblon ligand with PEG linker and terminal acid for onward chemistry
7259 TBK1 PROTAC® 3i Nov 2020
Potent TANK-binding kinase 1 (TBK1) Degrader
5927 NS 383 Nov 2020
ASIC blocker; active in vivo
7302 Sulfo-NHS-LC-Biotin Nov 2020
Amine reactive biotinylation reagent, cell impermeable
7260 TBK1 control PROTAC® 4 Nov 2020
Negative control for TBK1 PROTAC® 3i (Cat. No. 7259)
7198 JHU 37160 Nov 2020
High affinity and highly potent hM3Dq and hM4Di DREADD agonist; blood brain barrier penetrant
6322 LW 6 Nov 2020
Malate dehydrogenase-2 (MDH2) inhibitor; also inhibits HIF-1α
7294 VH 101 phenol-alkylC6-amine Oct 2020
VHL ligand with alkyl linker and terminal amine for onward chemistry
7357 PLpro inhibitor 6 Oct 2020
SARS-CoV and SARS-CoV-2 PLpro inhibitor
7199 (±)-Eriodictyol Oct 2020
Potent TRPV1 antagonist; also antioxidant; activates Nrf2/ARE signaling
7059 GLPG 0187 Oct 2020
Potent αv integrin inhibitor
7193 Deschloroclozapine Oct 2020
High affinity and highly potent activator of hM3Dq and hM4Di DREADDs; rapidly blood brain barrier penetrant
7350 Tocriscreen Antiviral Library Oct 2020
Antiviral compound library for high throughput screening, chemical biology applications and drug repurposing; contains 240 bioactive compounds (100 μL 10 mM DMSO solutions)
7329 Thalidomide 4'-ether-alkylC2-acid Oct 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7219 CRBN PROTAC® 14a Oct 2020
Cereblon Degrader
7188 Carfilzomib Oct 2020
Potent irreversible proteasome inhibitor; active in vivo
7106 VH 032 amide-alkylC2-acid Oct 2020
VHL ligand with alkyl linker and terminal acid for onward chemistry
7335 Thalidomide 4'-ether-alkylC8-acid Oct 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7331 Thalidomide 4'-ether-alkylC4-acid Oct 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7293 VH 101 phenol-alkylC4-amine Oct 2020
VHL ligand with alkyl linker and terminal amine for onward chemistry
7285 DCLK1-IN-1 Oct 2020
Potent and selective doublecortin like kinase 1/2 (DCLK1/2) inhibitor; orally bioavailable
7143 VX 765 Oct 2020
High affinity and selective caspase-4 and caspase 1/ICE inhibitor; orally bioavailable
5950 Ethyl LipotF Oct 2020
Selective FTO inhibitor
7330 Thalidomide 4'-ether-alkylC3-acid Sep 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7191 Santacruzamate A Sep 2020
Highly potent and selective HDAC2 inhibitor
6996 BOP-JF549 Sep 2020
Yellow fluorescent dual α9β1/α4β1 integrin inhibitor comprising BOP conjugated to Janelia Fluor® 549; fluorogenic; photostable
7287 FAM-DEALA-Hyp-YIPD Sep 2020
Fluorescent HIF-1α peptide; can be used to evaluate the effect of VHL binding on degradation activity
7334 Thalidomide 4'-ether-alkylC7-acid Sep 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7333 Thalidomide 4'-ether-alkylC6-acid Sep 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7332 Thalidomide 4'-ether-alkylC5-acid Sep 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7104 VH 032 amide-PEG1-acid Sep 2020
VHL ligand with PEG linker and terminal acid for onward chemistry
7279 Janelia Fluor® 646, Tetrazine Sep 2020
Red dye (Reactive group: tetrazine). Applications: super-resolution microscopy e.g. dSTORM & STED, confocal and live cell imaging
7277 HBC 530 Sep 2020
GFP fluorophore mimic for imaging RNA in live cells; activated by binding to Pepper aptamers; suitable for confocal and two-photon microscopy
6238 PKRA 7 Sep 2020
Potent prokineticin (PK) 1 and 2 receptor antagonist; antitumor; BBB penetrant
7298 xStAx-VHLL Sep 2020
Selective peptide-based β-catenin degrader
7095 Pomalidomide 4'-PEG5-acid Sep 2020
Cereblon ligand with PEG linker and terminal acid for onward chemistry
7262 SJF 1528 Sep 2020
Potent EGFR Degrader; also degrades HER2
7178 LCL 161, phenol Sep 2020
Functionalized IAP ligand for PROTACs
6913 Thalidomide 4'-oxyacetamide-alkylC1-PEG3-alkylC3-amine Sep 2020
Cereblon ligand with alkyl-PEG-alkyl linker and terminal amine for onward chemistry
7261 SJF 1521 Sep 2020
Selective EGFR Degrader
7288 Thalidomide-Cyanine 5 Sep 2020
Fluorescent cereblon probe
7076 Lenalidomide 4'-PEG3-amine Sep 2020
Cereblon ligand with PEG linker and terminal amine for onward chemistry
7075 Lenalidomide 4'-PEG1-amine Sep 2020
Cereblon ligand with PEG linker and terminal amine for onward chemistry
7159 FMF-04-159-R Sep 2020
Potent CDK14 and CDK16 inhibitor; displays reversible inhibition of CDK14
7158 FMF-04-159-2 Sep 2020
Potent covalent CDK14 and CDK16 inhibitor; also inhibits other TAIRE kinase family members
7283 Apilimod dimesylate Aug 2020
Potent and selective PIKfyve inhibitor
7170 D-GsMTx4 Aug 2020
TRPC1/6 and Piezo2 inhibitor; resistant to proteolytic digestion
6267 Taxol Janelia Fluor ® 549 Aug 2020
Yellow fluorescent taxol derivative; probe for microtubule staining
7187 Zanamivir Aug 2020
Potent influenza virus neuraminidase inhibitor
7091 Miro1 Reducer Aug 2020
Promotes mitochondrial Rho GTPase 1 (Miro1) degradation
7093 Lenalidomide 4'-PEG2-amine Aug 2020
Cereblon ligand with PEG linker and terminal amine for onward chemistry
7231 EIDD 1931 Aug 2020
Viral RNA-dependent RNA polymerase (RdRP) inhibitor; broad spectrum antiviral nucleotide
7209 Pomalidomide 4'-alkylC4-acid Aug 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
6916 dTAG-13-NEG Aug 2020
Negative control for dTAG-13 (Cat. No. 6605)
6915 dTAGV-1-NEG Aug 2020
Negative control for dTAGV-1 (Cat. No. 6914)
6914 dTAGV-1 Aug 2020
Potent and selective degrader of mutant FKBP12F36V fusion proteins
7280 GRL 0617 Aug 2020
Coronavirus PLpro inhibitor
7290 Famotidine Aug 2020
Potent and high affinity H2 biased inverse agonist
7029 GX 201 Aug 2020
Potent and selective Nav1.7 blocker; analgesic
6997 BOP-JF646 Aug 2020
Red fluorescent dual α9β1/α4β1 integrin inhibitor comprising BOP conjugated to Janelia Fluor® 646; fluorogenic; photostable
6297 AP 20187 Aug 2020
Chemical inducer of protein dimerization; active in vivo
7189 Saracatinib Aug 2020
Potent and selective Src tyrosine kinase family inhibitor; anticancer; antiviral; orally bioavailable
7212 Pomalidomide 4'-PEG2-acid Jul 2020
Cereblon ligand with PEG linker and terminal acid for onward chemistry
7270 iP300w Jul 2020
Potent p300/CBP inhibitor
6789 K 03861 Jul 2020
Potent Cdk2 inhibitor
7211 Pomalidomide 4'-alkylC8-acid Jul 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7272 dNTP solution mix Jul 2020
Mixture of deoxynucleotides for use in PCR
7108 VH 032 amide-alkylC8-acid Jul 2020
VHL ligand with alkyl linker and terminal acid for onward chemistry
7107 VH 032 amide-alkylC6-acid Jul 2020
VHL ligand with alkyl linker and terminal acid for onward chemistry
7094 Pomalidomide 4'-PEG1-acid Jul 2020
Cereblon ligand with PEG linker and terminal acid for onward chemistry
7230 MPro N3 Jul 2020
Coronavirus Mpro inhibitor
7087 AGI 5198 Jul 2020
Potent and selective inhibitor of mutant isocitrate dehydrogenase 1 (mIDH1)
7097 Pomalidomide 4'-alkylC7-acid Jul 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7160 DD 03-171 Jul 2020
Potent and selective BTK Degrader
6316 ASB 14780 Jul 2020
Potent and selective cytosolic phospholipase A2 alpha (cPLA2α) inhibitor; active in vivo; orally bioavailable
7210 Pomalidomide 4'-alkylC6-acid Jul 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
7204 Pomalidomide 4'-PEG3-amine Jul 2020
Cereblon ligand with PEG linker and terminal amine for onward chemistry
7203 Pomalidomide 4'-PEG1-amine Jul 2020
Cereblon ligand with PEG linker and terminal amine for onward chemistry
6943 dBRD9-A Jul 2020
Potent BRD9 Degrader
7235 Arbidol Jul 2020
Inhibits replication of SARS-CoV-2 in vitro; broad spectrum antiviral
7208 Pomalidomide 4'-alkylC7-amine Jul 2020
Cereblon ligand with alkyl linker and terminal amine for onward chemistry
7096 Pomalidomide 4'-alkylC3-acid Jul 2020
Cereblon ligand with alkyl linker and terminal acid for onward chemistry
6873 DC 271 Jul 2020
Fluorescent retinoic acid analog; solvochromatic probe
7224 Oseltamivir phosphate Jul 2020
Influenza virus neuraminidase inhibitor; antiviral prodrug
7234 Nitazoxanide Jul 2020
Pyruvate flavodoxin/ferredoxin oxidoreductase inhibitor; also inhibits Wnt signaling; broad spectrum anti-infective
6130 AP 1903 Jul 2020
Chemical inducer of protein dimerization; active in vivo
7220 A 410099.1 amide-PEG4-amine Jun 2020
IAP ligand with PEG linker and terminal amine for onward chemistry
7221 A 410099.1 amide-PEG5-amine Jun 2020
IAP ligand with PEG linker and terminal amine for onward chemistry
7001 AT 7867 Jun 2020
Potent pan-Akt and PKA inhibitor
6945 dBET6 Jun 2020
Potent and selective (+)-JQ1 based PROTAC targeting BET bromodomains, active in vivo
7227 GS 441524 Jun 2020
Viral RNA-dependent RNA polymerase (RdRP) inhibitor; broad spectrum antiviral nucelotide
7226 Remdesivir Jun 2020
Viral RNA-dependent RNA polymerase (RdRP) inhibitor; broad spectrum antiviral nucelotide prodrug
7081 LY 2886721 Hydrochloride Jun 2020
Potent and selective β-secretase (BACE) inhibitor
7056 Conduritol B epoxide Jun 2020
Irreversible glucocerebrosidase (β-glucosidase) inhibitor; used to generate Gaucher disease models
6391 CD38 inhibitor 78c Jun 2020
Potent CD38 inhibitor; active in vivo
7246 Nucleic Acid Dye Green I Jun 2020
High affinity double-stranded DNA (dsDNA) probe; used in RT-LAMP and qPCR
7232 SBP1-FITC Jun 2020
Fluorescent ACE2-derived peptide; binds receptor binding domain of SARS-CoV-2 spike protein
7052 Lopinavir Jun 2020
Highly potent and selective HIV-1 protease inhibitor
6430 Takinib Jun 2020
Potent and selective TAK1/MAP3K7 kinase inhibitor