Potent and selective PDE2A inhibitor (IC50 = 1 nM). Exhibits 2000-fold selectivity for PDE2A over PDE10A. Brain penetrant.
Sold for research purposes under agreement from Pfizer Inc.
|Storage||Store at -20°C|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
|Solvent||Max Conc. mg/mL||Max Conc. mM|
Preparing Stock Solutions
The following data is based on the product molecular weight 414.39. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||2.41 mL||12.07 mL||24.13 mL|
|5 mM||0.48 mL||2.41 mL||4.83 mL|
|10 mM||0.24 mL||1.21 mL||2.41 mL|
|50 mM||0.05 mL||0.24 mL||0.48 mL|
References are publications that support the products' biological activity.
If you know of a relevant reference for PF 05180999, please let us know.
View Related Products by Target
View Related Products by Product Action
Keywords: PF 05180999, supplier, PF05180999, potent, selective, phosphodiesterase, PDE, 2a, inhibitors, inhibits, brain, penetrant, Phosphodiesterases, Phosphodiesterases, Tocris Bioscience
Citations for PF 05180999
Citations are publications that use Tocris products.
Currently there are no citations for PF 05180999. Do you know of a great paper that uses PF 05180999 from Tocris? If so please let us know.
Reviews for PF 05180999
There are currently no reviews for this product. Be the first to review PF 05180999 and earn rewards!
Have you used PF 05180999?
Submit a review and receive an Amazon gift card.
$10US/$10CAN/€7/£6 gift card for a review without an image
$25US/$25CAN/€18/£15 gift card for a review with an image
*Offer only valid in the USA / Canada, UK and EuropeSubmit a Review