TGF-β Receptor Inhibitors

Cat. No. Product Name / Activity
6712 A 77-01
Potent inhibitor of TGF-βRI
2939 A 83-01
Selective inhibitor of TGF-βRI, ALK4 and ALK7
2902 D 4476
TGF-βRI inhibitor. Also inhibits CK1
6956 Galunisertib
ALK4 and ALK5 (TGFβRI) inhibitor
3264 GW 788388
Potent and selective inhibitor of TGF-βRI
6016 IN 1130
Potent and selective inhibitor of TGF-βRI
2718 LY 364947
Selective inhibitor of TGF-βRI
5288 R 268712
Potent and selective inhibitor of TGF-βRI
3742 RepSox
Potent and selective inhibitor of TGF-βRI
1614 SB 431542
Potent, selective inhibitor of TGF-βRI, ALK4 and ALK7
3263 SB 505124
Selective inhibitor of TGF-βRI, ALK4 and ALK7
3211 SB 525334
Selective inhibitor of TGF-βRI
3269 SD 208
Potent ATP-competitive TGF-βRI inhibitor
6245 SM 16
Potent TGF-βRI inhibitor; orally bioavailable