Nicotinic (α4β2) Receptor Modulators

Cat. No.	Product Name / Activity
5963	CMPI hydrochloride
	Potent positive allosteric modulator of α4β2 nAChRs; also inhibitor of (α4)₂(β2)₃, muscle-type and Torpedo nAChRs
3328	Desformylflustrabromine hydrochloride
	Positive allosteric modulator of α4β2 nAChRs; also muscle-type nAChR inhibitor
4141	LY 2087101
	Allosteric potentiator of α7, α4β2 and α4β4 nAChRs
5112	NS 9283
	Positive allosteric modulator of α4β2 nAChRs

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Literature in this Area

Nicotinic ACh Scientific Review

Nicotinic ACh Receptors Scientific Review

Our Nicotinic Acetylcholine Receptor review summarizes the structure and function of nAChR receptors, and the pharmacological ligands used to study them.

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Alzheimer's Life Science Poster

Written by Dimitra Sokolova and Soyon Hong

Our Alzheimer's disease poster summarizes the genetic, molecular and cellular changes observed in the progression of this neurodegenerative disease.

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