Nicotinic Receptors (Other Subtypes)
Nicotinic Receptor (Other Subtype) Agonists |
|
|---|---|
| Cat. No. | Product Name / Activity |
| 3549 | 3-Bromocytisine |
| Potent α4β4, α4β2 and α7 nAChR agonist | |
| 5236 | CC4 |
| High affinity and subtype-selective α6β2 and α4β2 nAChR partial agonist | |
| 4831 | NS 3861 |
| α3β2 full agonist; also α3β4 partial agonist | |
| 4766 | SIB 1508Y maleate |
| Potent agonist of α4β2, α2β4, α4β4 and α3β4 nACh receptors | |
Nicotinic Receptor (Other Subtype) Antagonists |
|
| Cat. No. | Product Name / Activity |
| 1340 | α-Conotoxin MII |
| Potent and selective α3β2 and β3 nAChR antagonist | |
| 2349 | Dihydro-β-erythroidine hydrobromide |
| α4β2, muscle type and Torpedo nAChR antagonist | |
| 4424 | SR 16584 |
| Selective α3β4 nAChR antagonist | |
Nicotinic Receptor (Other Subtype) Modulators |
|
| Cat. No. | Product Name / Activity |
| 3328 | Desformylflustrabromine hydrochloride |
| Muscle-type nAChR inhibitor; also positive allosteric modulator of α4β2 nAChRs | |
| 4141 | LY 2087101 |
| Allosteric potentiator of α7, α4β2 and α4β4 nAChRs | |
Nicotinic Receptor (Other Subtype) Inhibitors |
|
| Cat. No. | Product Name / Activity |
| 5963 | CMPI hydrochloride |
| Inhibitor of (α4)2(β2)3, muscle-type and Torpedo nAChRs; also potent positive allosteric modulator of α4β2 nAChRs | |
Nicotinic ACh Scientific Review
Our Nicotinic Acetylcholine Receptor review summarizes the structure and function of nAChR receptors, and the pharmacological ligands used to study them.
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