Agonists |
Cat. No. | Product Name / Activity |
---|---|
3549 | 3-Bromocytisine |
Potent α4β4, α4β2 and α7 nAChR agonist | |
5236 | CC4 |
High affinity and subtype-selective α6β2 and α4β2 nAChR partial agonist | |
1518 | 5-Iodo-A-85380 dihydrochloride |
High affinity α4β2 and α6β2 subtype-selective nAChR agonist | |
1527 | 5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative |
Precursor to 5-Iodo-A-85380 (Cat. No. 1518) | |
4831 | NS 3861 |
α3β2 full agonist; also α3β4 partial agonist | |
4766 | SIB 1508Y maleate |
Potent agonist of α4β2, α2β4, α4β4 and α3β4 nACh receptors | |
4764 | SIB 1553A hydrochloride |
nAChR agonist; displays selectivity for β4 subunit-containing receptors | |
1348 | UB 165 fumarate |
Subunit selective nAChR agonist | |
Antagonists |
Cat. No. | Product Name / Activity |
3120 | α-Conotoxin AuIB |
Selective α3β4 nAChR antagonist | |
1340 | α-Conotoxin MII |
Potent and selective α3β2 and β3 nAChR antagonist | |
3121 | α-Conotoxin PIA |
Selective antagonist of α6-containing nAChRs | |
3123 | α-Conotoxin PnIA |
Selective α3β2 nAChR antagonist | |
2349 | Dihydro-β-erythroidine hydrobromide |
α4β2, muscle type and Torpedo nAChR antagonist | |
4424 | SR 16584 |
Selective α3β4 nAChR antagonist | |
Modulators |
Cat. No. | Product Name / Activity |
3328 | Desformylflustrabromine hydrochloride |
Muscle-type nAChR inhibitor; also positive allosteric modulator of α4β2 nAChRs | |
4141 | LY 2087101 |
Allosteric potentiator of α7, α4β2 and α4β4 nAChRs | |
Inhibitors |
Cat. No. | Product Name / Activity |
5963 | CMPI hydrochloride |
Inhibitor of (α4)2(β2)3, muscle-type and Torpedo nAChRs; also potent positive allosteric modulator of α4β2 nAChRs |