κ Opioid Receptor Agonists

Cat. No. Product Name / Activity
3195 Dynorphin A
Endogenous κ agonist
1483 GR 89696 fumarate
Subtype-selective κ agonist
0822 ICI 204,448 hydrochloride
κ agonist, acts peripherally
8135 PIPE 3297 dihydrochloride
Potent and selective κ opioid receptor agonist; devoid of β-Arrestin-2 recruitment. Also induces differentiation of OPC.
0471 (+)-U-50488 hydrochloride
Selective κ agonist; less active enantiomer of (±)-U-50488 (Cat. No. 0495)
0495 (±)-U-50488 hydrochloride
Selective κ agonist
0496 (-)-U-50488 hydrochloride
Selective κ agonist; more active enantiomer of (±)-U-50488 (Cat. No. 0495)