EGFR Inhibitors

Cat No Product Name / Activity
5318 AEE 788
Potent EGFR and VEGFR inhibitor
1276 AG 1478 hydrochloride
Highly potent EGFR-kinase inhibitor
0493 AG 18
EGFR/PDGFR-kinase inhibitor
0414 AG 490
EGFR-kinase inhibitor. Also JAK2, JAK3 inhibitor
0619 AG 494
Potent EGFR-kinase inhibitor
0618 AG 555
Potent EGFR-kinase inhibitor
0616 AG 556
EGFR-kinase inhibitor
1555 AG 825
Selective ErbB2 inhibitor
2617 AG 879
ErbB2 inhibitor
0497 AG 99
EGFR-kinase inhibitor
4397 AV 412
Potent inhibitor of EGFR, ErbB2 and Abl receptor tyrosine kinases
2417 BIBU 1361 dihydrochloride
Selective inhibitor of EGFR-kinase
2416 BIBX 1382 dihydrochloride
Highly selective EGFR-kinase inhibitor
5022 BMS 599626 dihydrochloride
Potent, selective EGFR and ErbB2 inhibitor
5916 Canertinib dihydrochloride
Potent EGFR kinase inhibitor
3360 CGP 52411
EGFR inhibitor. Also inhibits Aβ42 fibril formation
5973 CP 724714
Potent and selective ErbB2 inhibitor
6231 Dacomitinib
Potent irreversible pan ErbB inhibitor
4502 DIM
Inhibits EGFR activation; also induces apoptosis
1110 Genistein
EGFR kinase inhibitor. Also estrogen and PPARγ ligand
2239 GW 583340 dihydrochloride
Potent dual EGFR/ErbB2 inhibitor; orally active
3580 HKI 357
Dual irreversible inhibitor of ErbB2 and EGFR
3000 Iressa
Orally active, selective EGFR inhibitor
3352 JNJ 28871063 hydrochloride
Potent ErbB receptor family inhibitor
1331 Lavendustin A
EGFR, p60c-src inhibitor
0577 Methyl 2,5-dihydroxycinnamate
EGFR-kinase inhibitor
1037 PD 153035 hydrochloride
EGFR-kinase inhibitor
2615 PD 158780
Potent ErbB receptor family inhibitor
5939 PF 6274484
High affinity and potent covalent EGFR kinase inhibitor
4941 PKI 166 hydrochloride
Potent EGFR-kinase inhibitor
2794 PP 3
EGFR-kinase inhibitor. Also Src kinase negative control
3599 TAK 165
Potent and selective ErbB2 inhibitor
0578 Tyrphostin B44, (-) enantiomer
EGFR-kinase inhibitor
0579 Tyrphostin B44, (+) enantiomer
EGFR-kinase inhibitor
3115 WHI-P 154
Potent EGFR inhibitor. Also inhibits JAK3