Cat. No. | Product Name / Activity |
---|---|
5584 | Aripiprazole |
High affinity D2 and 5-HT1A partial agonist; also 5-HT2A antagonist | |
3346 | ATC 0175 hydrochloride |
5-HT1A partial agonist; also 5-HT2B antagonist and MCH1 antagonist | |
1006 | BMY 7378 dihydrochloride |
5-HT1A partial agonist | |
0556 | BP 554 maleate |
Selective 5-HT1A agonist | |
0962 | Buspirone hydrochloride |
5-HT1A partial agonist | |
1080 | (R)-(+)-8-Hydroxy-DPAT hydrobromide |
Selective 5-HT1A agonist; enantiomer of 8-Hydroxy-DPAT hydrobromide (Cat. No. 0529) | |
0529 | 8-Hydroxy-DPAT hydrobromide |
Selective 5-HT1A agonist; also has moderate affinity for 5-HT7 | |
0797 | 8-Hydroxy-PIPAT oxalate |
High affinity 5-HT1A agonist | |
1869 | Ipsapirone |
Selective 5-HT1A agonist | |
0411 | MDL 73005EF hydrochloride |
Potent and selective 5-HT1A partial agonist | |
1746 | Nemonapride |
5-HT1A agonist; also highly potent D2-like dopamine antagonist | |
0912 | RU 24969 hemisuccinate |
5-HT1A and 5-HT1B agonist | |
1771 | S 14506 hydrochloride |
Highly potent 5-HT1A agonist; displays unique binding mechanism | |
2854 | Tandospirone hydrochloride |
Selective 5-HT1A partial agonist | |
1772 | Urapidil hydrochloride |
5-HT1A agonist; also α1-adrenoceptor antagonist | |
6202 | Vilazodone hydrochloride |
Potent 5-HT1A partial agonist and SSRI; antidepressant | |
2491 | Xaliproden hydrochloride |
High affinity 5-HT1A agonist; orally active |