5-HT1A Receptor Agonists

Cat. No. Product Name / Activity
5584 Aripiprazole
High affinity D2 and 5-HT1A partial agonist; also 5-HT2A antagonist
3346 ATC 0175 hydrochloride
5-HT1A partial agonist; also 5-HT2B antagonist and MCH1 antagonist
1006 BMY 7378 dihydrochloride
5-HT1A partial agonist
0556 BP 554 maleate
Selective 5-HT1A agonist
0962 Buspirone hydrochloride
5-HT1A partial agonist
1080 (R)-(+)-8-Hydroxy-DPAT hydrobromide
Selective 5-HT1A agonist; enantiomer of 8-Hydroxy-DPAT hydrobromide (Cat. No. 0529)
0529 8-Hydroxy-DPAT hydrobromide
Selective 5-HT1A agonist; also has moderate affinity for 5-HT7
0797 8-Hydroxy-PIPAT oxalate
High affinity 5-HT1A agonist
1869 Ipsapirone
Selective 5-HT1A agonist
0411 MDL 73005EF hydrochloride
Potent and selective 5-HT1A partial agonist
1746 Nemonapride
5-HT1A agonist; also highly potent D2-like dopamine antagonist
0912 RU 24969 hemisuccinate
5-HT1A and 5-HT1B agonist
1771 S 14506 hydrochloride
Highly potent 5-HT1A agonist; displays unique binding mechanism
2854 Tandospirone hydrochloride
Selective 5-HT1A partial agonist
1772 Urapidil hydrochloride
5-HT1A agonist; also α1-adrenoceptor antagonist
6202 Vilazodone hydrochloride
Potent 5-HT1A partial agonist and SSRI; antidepressant
2491 Xaliproden hydrochloride
High affinity 5-HT1A agonist; orally active