GPBA Receptors

More Information »GPBA receptors (TGR5, GPBAR1, M-BAR) are G protein-coupled receptors (GPCRs) that are activated by bile acids. They are highly expressed in the gallbladder, ileum and colon, and are important in the regulation of glucose and lipid metabolism, and energy utilization.

GPBA Receptor Products

Agonists
Cat.No.
Product Name / Activity
3906 Betulinic acid
Antitumor and anti-HIV agent; GPBA receptor (TGR5) agonist; also activates NF-κB
4478 GPBAR-A
GPBA receptor (TGR5) agonist
6026 Oleanolic acid
Selective GPBA receptor (TGR5) partial agonist
5129 TC-G 1005
Potent and selective GPBA receptor (TGR5) agonist
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