Other Nuclear Receptors

Agonists

Cat No Product Name / Activity
5459 Cytosporone B
High affinity Nur77 agonist
6376 DIM-C-pPhOCH3
Nur77 agonist
4378 DLPC
Selective liver receptor homolog-1 (LRH-1) agonist
4554 GC 1
High affinity thyroid receptor α (TRα) and TRβ agonist; thyromimetic

Antagonists

Cat No Product Name / Activity
3043 AC 45594
SF-1 inverse agonist
4957 ML 179
Selective liver receptor homolog 1 (LRH1) inverse agonist
3440 SID 7969543
Selective steroidogenic factor-1 (SF-1, NR5A1) inhibitor

Activators

Cat No Product Name / Activity
5821 C-DIM 12
Nurr1 activator; inhibits NF-κB-dependent gene expression
5699 IP7e
Potent Nurr1 activator

Other

Cat No Product Name / Activity
2013 Guggulsterone
Broad spectrum steroid receptor ligand. Antagonizes FXR and displays hypolipidemic activity
3570 Z-Guggulsterone
Broad spectrum steroid receptor ligand. More active isomer of guggulsterone (Cat. No. 2013)
5552 Liothyronine sodium
Thyroid hormone (T3) analog; also promotes adipogenic differentiation of MSCs
5964 SI-2 hydrochloride
Steroid receptor coactivator 3 (SRC-3) inhibitor