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Other Nuclear Receptors

Agonists
Cat. No. Product Name / Activity
4554 GC 1
High affinity thyroid receptor α (TRα) and TRβ agonist; thyromimetic

Inverse Agonists
Cat. No. Product Name / Activity
3043 AC 45594
SF-1 inverse agonist
4957 ML 179
Selective liver receptor homolog 1 (LRH1) inverse agonist

Antagonists
Cat. No. Product Name / Activity
3440 SID 7969543
Selective steroidogenic factor-1 (SF-1, NR5A1) inhibitor

Degraders
Cat. No. Product Name / Activity
7388 ND1-YL2
SRC-1 peptide-based Degrader; active in vivo

Other
Cat. No. Product Name / Activity
2013 Guggulsterone
Broad spectrum steroid receptor ligand. Antagonizes FXR and displays hypolipidemic activity
3570 Z-Guggulsterone
Broad spectrum steroid receptor ligand. More active isomer of guggulsterone (Cat. No. 2013)
5964 SI-2 hydrochloride
Steroid receptor coactivator 3 (SRC-3) inhibitor
6666 T3
Thyroid hormone; also promotes differentiation of oligodendroglial precursor cells