Nicotinic (α4β2) Receptor Agonists
| Cat. No. | Product Name / Activity |
|---|---|
| 5079 | ABT 089 dihydrochloride |
| High affinity and selective α4β2 nAChR partial agonist | |
| 6576 | ABT 594 hydrochloride |
| Selective α4β2 nAChR agonist | |
| 3549 | 3-Bromocytisine |
| Potent α4β4, α4β2 and α7 nAChR agonist | |
| 5236 | CC4 |
| High affinity and subtype-selective α6β2 and α4β2 nAChR partial agonist | |
| 3546 | (-)-Nicotine ditartrate |
| Prototypical nAChR agonist | |
| 1053 | RJR 2403 oxalate |
| Selective α4β2 nAChR agonist | |
| 2737 | TC 2559 difumarate |
| Selective α4β2 nAChR partial agonist | |
| 6865 | uPSEM 792 hydrochloride |
| α4β2 partial agonist; uPSEM agonist for PSAM4-GlyR and PSAM4-5HT3; brain-penetrant | |
| 3754 | Varenicline tartrate |
| Selective α4β2 nAChR partial agonist; orally active |

