Nicotinic (α4β2) Receptor Agonists

Cat. No. Product Name / Activity
5017 A 85380 dihydrochloride
High affinity and selective α4β2 nAChR agonist
5079 ABT 089 dihydrochloride
High affinity and selective α4β2 nAChR partial agonist
6576 ABT 594 hydrochloride
Selective α4β2 nAChR agonist
3549 3-Bromocytisine
Potent α4β4, α4β2 and α7 nAChR agonist
5236 CC4
High affinity and subtype-selective α6β2 and α4β2 nAChR partial agonist
3546 (-)-Nicotine ditartrate
Prototypical nAChR agonist
1053 RJR 2403 oxalate
Selective α4β2 nAChR agonist
2737 TC 2559 difumarate
Selective α4β2 nAChR partial agonist
6865 uPSEM 792 hydrochloride
α4β2 partial agonist; uPSEM agonist for PSAM4-GlyR and PSAM4-5HT3; brain-penetrant
3754 Varenicline tartrate
Selective α4β2 nAChR partial agonist; orally active