Nicotinic (α4β2) Receptor Agonists

Cat. No. Product Name / Activity
5017 A 85380 dihydrochloride
High affinity and selective α4β2 nAChR agonist
5079 ABT 089 dihydrochloride
High affinity and selective α4β2 nAChR partial agonist
6576 ABT 594 hydrochloride
Selective α4β2 nAChR agonist
3549 3-Bromocytisine
Potent α4β4, α4β2 and α7 nAChR agonist
5236 CC4
High affinity and subtype-selective α6β2 and α4β2 nAChR partial agonist
5557 Dianicline
Selective α4β2 nAChR partial agonist
6706 DPNB-ABT 594
Caged ABT 594 (Cat. No. 6576); suitable for one- or two-photon photolysis
1518 5-Iodo-A-85380 dihydrochloride
High affinity α4β2 and α6β2 subtype-selective nAChR agonist
1527 5-Iodo-A-85380, 5-trimethylstannyl N-BOC derivative
Precursor to 5-Iodo-A-85380 (Cat. No. 1518)
3546 (-)-Nicotine ditartrate
Prototypical nAChR agonist
1053 RJR 2403 oxalate
Selective α4β2 nAChR agonist
4766 SIB 1508Y maleate
Potent agonist of α4β2, α2β4, α4β4 and α3β4 nACh receptors
2737 TC 2559 difumarate
Selective α4β2 nAChR partial agonist
6865 uPSEM 792 hydrochloride
α4β2 partial agonist; uPSEM agonist for PSAM4-GlyR and PSAM4-5HT3; brain-penetrant
3754 Varenicline tartrate
Selective α4β2 nAChR partial agonist; orally active