Inward Rectifier Potassium (Kir) Channel Blockers
| Cat. No. | Product Name / Activity |
|---|---|
| 6086 | AMP PNP |
| Kir6 blocker; non-hydrolyzable AMP analog | |
| 1513 | CGP 7930 |
| Blocks G protein-coupled inwardly rectifying K+ (GIRK) channels | |
| 0911 | Glibenclamide |
| Kir6 (KATP) channel blocker | |
| 4549 | ML 133 hydrochloride |
| Kir2 channel blocker | |
| 6889 | ML 418 |
| Kir 7.1 inhibitor; also inhibits Kir 6.2 | |
| 4231 | Nateglinide |
| Kir6 (KATP) blocker; displays high affinity for SUR1/Kir6.2 channels | |
| 3805 | Repaglinide |
| Kir6 (KATP) channel blocker | |
| 0925 | SCH 23390 hydrochloride |
| Kir3 channel blocker; also potent dopamine D1-like antagonist and 5-HT2C agonist | |
| 3948 | Terfenadine |
| KV11.1 (hERG) and Kir6 (KATP) channel blocker. Also H1 antagonist | |
| 1316 | Tertiapin-Q |
| Selective blocker of inward-rectifier K+ channels | |
| 6877 | VU 0134992 |
| Kir4.1 blocker | |
| 8151 | VU 0542270 |
| Selective inhibitor of Kir6.1 KATP channels |