Inward Rectifier Potassium (Kir) Channel Blockers

Cat. No. Product Name / Activity
6086 AMP PNP
Kir6 blocker; non-hydrolyzable AMP analog
0911 Glibenclamide
Kir6 (KATP) channel blocker
4549 ML 133 hydrochloride
Kir2 channel blocker
6889 ML 418
Kir 7.1 inhibitor; also inhibits Kir 6.2
4231 Nateglinide
Kir6 (KATP) blocker; displays high affinity for SUR1/Kir6.2 channels
2095 PNU 37883 hydrochloride
Vascular Kir6 (KATP) channel blocker
3805 Repaglinide
Kir6 (KATP) channel blocker
0925 SCH 23390 hydrochloride
Kir3 channel blocker; also potent dopamine D1-like antagonist and 5-HT2C agonist
3948 Terfenadine
KV11.1 (hERG) and Kir6 (KATP) channel blocker. Also H1 antagonist
1316 Tertiapin-Q
Selective blocker of inward-rectifier K+ channels
6877 VU 0134992
Kir4.1 blocker