GABAA Receptor Benzodiazepines

Cat. No. Product Name / Activity
3568 Bretazenil
Benzodiazepine partial agonist
0405 β-CCB
Benzodiazepine inverse agonist; putative endogenous ligand
2467 CGS 20625
Selective benzodiazepine partial agonist
0456 Chlormezanone
Positive allosteric modulator of benzodiazepine site
1709 CL 218872
Benzodiazepine agonist
2805 Diazepam
Acts at the benzodiazepine modulatory site
0505 Dihydroergotoxine mesylate
Binds to GABAA receptor Cl- channel; allosteric modulator of benzodiazepine site
3083 DMCM hydrochloride
Benzodiazepine inverse agonist
0554 FG 7142
Benzodiazepine inverse agonist
0658 FGIN-1-27
Potent ligand for mitochondrial DBI receptor; GABAA receptor modulator
0659 FGIN-1-43
Potent ligand for mitochondrial DBI receptor; GABAA receptor modulator
1328 Flumazenil
Benzodiazepine antagonist
2174 Hispidulin
Partial positive allosteric modulator at the benzodiazepine site
3597 Indiplon
Positive allosteric modulator of GABAA; acts at benzodiazepine site
1327 L-655,708
Benzodiazepine inverse agonist; selective for α5-containing GABAA receptors
2832 Midazolam hydrochloride
Benzodiazepine agonist
1997 Ro 15-4513
Benzodiazepine partial inverse agonist
3942 TCS 1105
GABAA α2 benzodiazepine agonist
4414 TP 003
GABAA partial agonist; acts at benzodiazepine site
1994 ZK 93423 hydrochloride
Potent benzodiazepine agonist
1996 ZK 93426 hydrochloride
Potent and competitive benzodiazepine antagonist