5-HT2A Receptor Antagonists

Cat No Product Name / Activity
1809 Altanserin hydrochloride
5-HT2A receptor antagonist
5584 Aripiprazole
5-HT2A antagonist; also D2 and 5-HT1A receptor partial agonist
4468 AT 1015
Long-acting 5-HT2A antagonist
0444 Clozapine
5-HT2A and 5-HT2C antagonist; also dopamine antagonist
4480 DV 7028 hydrochloride
Selective 5-HT2A antagonist; antithrombotic
4470 EMD 281014 hydrochloride
Selective 5-HT2A antagonist
4958 Eplivanserin hemifumarate
Potent and selective 5-HT2A antagonist
0523 4F 4PP oxalate
Selective 5-HT2A antagonist
2645 Fananserin
5-HT2A antagonist; also D4 antagonist
0908 Ketanserin tartrate
Selective 5-HT2A antagonist. Also antagonist at 5-HT1D
4173 MDL 100907
Potent and selective 5-HT2A antagonist
0870 MDL 11,939
5-HT2A antagonist
2495 Melperone hydrochloride
5-HT2A/D2 receptor antagonist; neuroleptic
1644 Mesulergine hydrochloride
5-HT2A and 5-HT2C antagonist; also dopamine receptor partial agonist
2777 Nefazodone hydrochloride
5-HT2A antagonist; also 5-HT uptake inhibitor; antidepressant
4493 Paliperidone
Atypical antipsychotic; 5-HT2A and D2 antagonist
2735 PNU 96415E
5-HT2A and D4 antagonist; antipsychotic
1742 R-96544 hydrochloride
Potent, selective 5-HT2A antagonist
2865 Risperidone
5-HT2A antagonist
3739 Sarpogrelate hydrochloride
Selective 5-HT2A antagonist
0995 Spiperone hydrochloride
5-HT2A antagonist; also D2-like antagonist
6336 Trazodone hydrochloride
5-HT2A and α1 adrenoceptor antagonist; also enhances neural differentiation; antidepressant and neuroprotectant
3085 Ziprasidone hydrochloride
5-HT2A/D2 antagonist; atypical antipsychotic
3996 Zotepine
5-HT2A/D2 antagonist; atypical antipsychotic