Post-Translational Modification Inhibitors

Cat. No. Product Name / Activity
3084 Anacardic acid
Inhibits SUMOylation; also inhibits histone acetyltransferase
1744 Bay 11-7821
E2 ubiquitin (Ub) conjugating enzymes inhibitor
4200 C 646
Selective p300/CBP inhibitor
4503 CC 0651
Allosteric inhibitor of hCdc34
3416 Tris DBA
N-myristoyltransferase-1 inhibitor; antiproliferative
5646 EML 425
Reversible and non-competitive p300/CBP inhibitor
2407 FTI 277
Prodrug form of FTI 276 (Cat. No. 2406)
2430 GGTI 298
Geranylgeranyltransferase I (GGTase I) inhibitor
6326 Ginkgolic Acid
Inhibitor of SUMOylation
2637 Gliotoxin
Farnesyltransferase and geranylgeranyltransferase I inhibitor
5045 L002
p300 inhibitor
6265 Lonafarnib
Potent farnesyl transferase inhibitor
5103 Lys-CoA
Selective p300 inhibitor
4993 NSC 624206
Ubiquitin-activating enzyme (E1) inhibitor
4858 NSC 697923
Selective UBE2N inhibitor
4903 NU 9056
Inhibitor of KAT5 (Tip60) histone acetyltransferase
2978 PYR 41
Ubiquitin-activating enzyme (E1) inhibitor
4994 PYZD 4409
Ubiquitin-activating enzyme (E1) inhibitor
6410 Tipifarnib
Potent farnesyltransferase inhibitor; orally bioavailable