Post-Translational Modification Inhibitors

Cat. No. Product Name / Activity
3084 Anacardic acid
Inhibits SUMOylation; also inhibits histone acetyltransferase
1744 Bay 11-7821
E2 ubiquitin (Ub) conjugating enzymes inhibitor
4200 C 646
p300/CBP inhibitor
7907 DC 432
Potent peptidomimetic inhibitor of N-terminal methyltransferase 1/2
5646 EML 425
Reversible and non-competitive p300/CBP inhibitor
2430 GGTI 298
Geranylgeranyltransferase I (GGTase I) inhibitor
6265 Lonafarnib
Potent farnesyl transferase inhibitor
4993 NSC 624206
Ubiquitin-activating enzyme (E1) inhibitor
4903 NU 9056
Inhibitor of KAT5 (Tip60) histone acetyltransferase
2978 PYR 41
Ubiquitin-activating enzyme (E1) inhibitor