Multidrug Transporter Substrates
| Cat. No. | Product Name / Activity |
|---|---|
| 5119 | Calcein AM |
| Substrate for MDR | |
| 4936 | Clozapine N-oxide (CNO) |
| Metabolite of clozapine (Cat. No. 0444); shown to be a P-gp efflux pump substrate | |
| 6329 | Clozapine N-oxide dihydrochloride |
| Water soluble salt of Clozapine N-oxide (Cat. No. 4936); shown to be a P-gp efflux pump substrate | |
| 4054 | PEP 005 |
| Substrate for MDR; also protein kinase C activator |
