Multidrug Transporter Inhibitors

Cat. No. Product Name / Activity
5867 Ceefourin 1
Selective MRP4 inhibitor
4193 CP 100356 hydrochloride
P-gp inhibitor
4646 Elacridar hydrochloride
P-gp inhibitor
2876 Fumitremorgin C
Inhibitor of BCRP-mediated multidrug resistance
3241 Ko 143
Potent and selective BCRP inhibitor
4169 KS 176
Selective BCRP inhibitor
2338 MK 571
MRP1 inhibitor; also CysLT1 (LTD4) inverse agonist
4107 Probenecid
MRP and OAT3 inhibitor
2775 Probucol
ABCA1 (CERP) inhibitor; also antioxidant, anti-inflammatory and hypocholesterolemic agent
4042 PSC 833
Inhibitor of P-gp-mediated MDR
6885 PU 23
Multidrug resistance protein (MRP) 4 inhibitor
3918 Pyrimethamine
Potent inhibitor of multidrug and toxin extrusion (MATE) transporters; also DHFR and STAT3 inhibitor
3722 Reversan
Selective MRP1 and P-gp inhibitor
5757 Tariquidar dihydrochloride
Potent P-glycoprotein (P-gp) inhibitor
5456 Zosuquidar trihydrochloride
High affinity P-gp inhibitor