| Cat. No. |
Product Name / Activity |
| 0414 |
AG 490 |
| JAK2, JAK3 inhibitor. Also EGFR-kinase inhibitor |
| 5617 |
AZD 1480 |
| Potent and selective JAK2 inhibitor; antiangiogenic |
| 7222 |
Baricitinib |
| Highly potent JAK1 and JAK2 inhibitor; also inhibits JAK3 and Tyk2 |
| 4500 |
Cercosporamide |
| Potent Mnk2 inhibitor; also inhibits JAK3 |
| 4556 |
CP 690550 citrate |
| Potent JAK inhibitor |
| 1571 |
Cucurbitacin I |
| Selective inhibitor of STAT3/JAK2 signaling |
| 3395 |
Lestaurtinib |
| JAK2, FLT3 and TrkA inhibitor; also inhibits AurA and AurB |
| 6506 |
PF 06551600 malonate |
| Potent and selective JAK3 inhibitor |
| 6577 |
Pyridone 6 |
| Potent pan-JAK inhibitor; induces intermediate mesoderm; cell-permeable |
| 7064 |
Ruxolitinib |
| Potent and selective JAK1/JAK2 inhibitor; orally bioavailable |
| 7048 |
Ruxolitinib phosphate |
| Phosphate salt of Ruxolitinib (Cat. No. 7064); potent and selective JAK1/JAK2 inhibitor |
| 3035 |
SD 1008 |
| JAK2/STAT3 signaling pathway inhibitor |
| 6125 |
TC JL 37 |
| Potent TYK2 inhibitor |
| 7783 |
Upadacitinib |
| JAK1-selective inhibitor |