Heterotrimeric G-protein GTPase Inhibitors

Cat. No. Product Name / Activity
5642 CMPD101
Potent and selective GRK2/3 inhibitor
5245 Ebselen
Selectively inhibits Gq protein signaling
3090 Gallein
Inhibitor of Gβ/γ signaling
3594 GRK2i
GRK2 inhibitory polypeptide; Gβ/γ antagonist
1240 NF 023
Inhibitor of Go/i α-subunits; also P2X1 purinoceptor antagonist
1400 SCH 202676 hydrobromide
Inhibitor of ligand binding to G-protein-coupled receptors
7352 YM 254890
Gα-protein inhibitor; potent inhibitor of Gq/11 signaling