ETB Receptors
The endothelinB receptor (ETB receptor) is a member of the endothelin receptor group of G-protein-coupled receptors that also includes ETA. They are located primarily in vascular endothelial cells where they play a role in vasoconstriction, vasodilation and cell proliferation.
ETB Receptor Agonists |
|
|---|---|
| Cat. No. | Product Name / Activity |
| 1189 | BQ-3020 |
| Selective ETB agonist | |
| 1196 | IRL-1620 |
| Highly selective ETB agonist | |
| 1175 | Sarafotoxin S6c |
| Selective ETB agonist | |
ETB Receptor Antagonists |
|
| Cat. No. | Product Name / Activity |
| 1500 | BQ 788 sodium salt |
| Selective ETB antagonist | |
| 1838 | IRL-2500 |
| Potent ETB antagonist | |
The endothelinB receptor (ETB receptor) is a member of the endothelin receptor group of G-protein-coupled receptors that also includes ETA. They are located primarily in the vascular endothelial cells where they play a role in vasoconstriction, vasodilation, bronchoconstriction and cell proliferation. The human ETB receptor gene has been localized to chromosome 13 (13q22).