Cytochrome P450 Inhibitors

Cat. No. Product Name / Activity
6520 Abiraterone acetate
Potent CYP17A1 inhibitor
5038 ABT
Cytochrome P450 inhibitor; inhibits 20-HETE synthesis
3388 Anastrozole
Potent aromatase (CYP19) inhibitor
6170 Cinacalcet hydrochloride
Potent CYP2D2 inhibitor; also CaSR allosteric agonist and Ca2+ channel blocker
4096 Clotrimazole
Cytochrome P450 inhibitor; antifungal
3759 Exemestane
Steroidal aromatase (CYP19) inhibitor
6108 Galeterone
CYP17 inhibitor; also androgen receptor antagonist
1103 Ketoconazole
Cytochrome P450c17 inhibitor
4382 Letrozole
Potent, reversible non-steroidal aromatase inhibitor
2705 Liarozole dihydrochloride
Cytochrome P450 (CYP26) inhibitor; blocks retinoic acid metabolism
3292 Metyrapone
Cytochrome P450 inhibitor
2583 Omeprazole
CYP2C19, CYP2C9 and CYP3A inhibitor. Also H+,K+-ATPase inhibitor
4252 PF 4981517
Selective CYP3A4 inhibitor
1509 TMS
Cytochrome P450 1B1 inhibitor
5680 Vatalanib succinate
Potent aromatase inhibitor; also VEGFR inhibitor
3278 YM 511
Potent aromatase (CYP19) inhibitor