Casein Kinase 1 Inhibitors

Cat. No. Product Name / Activity
5329 CKI 7 dihydrochloride
CK1 inhibitor
3605 (R)-CR8
CK1 inhibitor; also potently inhibits cdk1 and cdk2
2902 D 4476
Selective CK1 inhibitor. Also inhibits TGF-βRI
3610 (R)-DRF053 dihydrochloride
Potent CK1 inhibitor; also inhibits cyclin-dependent kinases
6340 Epiblastin A
CK1 inhibitor; converts epiblast stem cells to ESCs and promotes ESC self-renewal
6676 IC 261
CK1 inhibitor; displays selectivity for CK1δ and CK1ε
4896 LH 846
Selective casein kinase 1δ inhibitor
4281 PF 4800567 hydrochloride
Selective casein kinase 1ε inhibitor
6346 PF 5006739
Potent CK1δ/ε inhibitor
3316 PF 670462
Potent and selective CK1ε and CK1δ inhibitor
5767 SR 3029
Potent and selective CK1δ and CK1ε inhibitor
4254 TAK 715
Inhibitor of Wnt/β-catenin signaling; cross-reacts with CK1δ/ε