Melatonin Receptors

More Information »Melatonin receptors are a group of high affinity Gi/G0 protein-coupled receptors, which are split into two subtypes; MT1 and MT2. They are widely distributed with high concentrations found in the brain (especially in the suprachiasmatic nucleus) and in the retina.

Melatonin Receptor Products

Product Name / Activity
0357 N-Acetyltryptamine
Melatonin partial agonist (MT1/MT2). Also MT3 antagonist
0443 6-Chloromelatonin
Melatonin agonist
0737 2-Iodomelatonin
High affinity melatonin agonist
3550 Melatonin
Endogenous hormone; agonist at MT1 and MT2
1035 8-M-PDOT
Melatonin agonist
0680 2-Phenylmelatonin
Potent melatonin agonist
Product Name / Activity
1218 DH 97
MT2 receptor antagonist
0877 Luzindole
Competitive melatonin MT1/MT2 antagonist
1034 4-P-PDOT
MT2 antagonist
0623 Prazosin hydrochloride
MT3 antagonist, also α1 and α2B antagonist
Product Name / Activity
0896 GR 135531
High affinity melatonin MT3 ligand

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