Histamine H1 Receptor Antagonists
| Cat. No. | Product Name / Activity |
|---|---|
| 3489 | Astemizole |
| Orally active, potent H1 antagonist; also KV11.1 (hERG) channel blocker | |
| 1453 | Clemastine fumarate |
| H1 antagonist | |
| 1425 | (S)-(+)-Dimethindene maleate |
| H1 antagonist. Also M2 muscarinic antagonist | |
| 3072 | Diphenhydramine hydrochloride |
| H1 antagonist | |
| 4245 | Meclizine dihydrochloride |
| H1 antagonist; human pregnane X receptor agonist | |
| 2018 | Mirtazapine |
| Potent H1 antagonist; also 5-HT2, 5-HT3 and α2 antagonist; antidepressant | |
| 4241 | Olopatadine hydrochloride |
| H1 antagonist; ocular antiallergic agent | |
| 3948 | Terfenadine |
| H1 antagonist. Also KV11.1 (hERG) and Kir6 (KATP) channel blocker |
Histamine Scientific Review
Our Histamine review gives an overview of the different histamine receptor subtypes, as well as highlighting pharmacological ligands for their study.
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