Estrogen (GPER) Receptors

More Information »The GPER (G protein-coupled estrogen receptor, GPR30) is a membrane protein that binds estrogen leading to estrogen-mediated adenylyl cyclase stimulation. The receptor is widely distributed in neural, breast, placental, heart, ovarian, prostate and hepatic tissues.

Estrogen (GPER) Receptor Products

Product Name / Activity
2824 β-Estradiol
Endogenous ER agonist
3577 G-1
Potent and selective GPER agonist
1110 Genistein
GPER agonist. Also tyrosine kinase inhibitor
1047 ICI 182,780
High affinity GPER agonist
1125 Quercetin
GPER agonist. Also non-selective PI 3-kinase inhibitor
0999 Tamoxifen citrate
High affinity GPER agonist
Product Name / Activity
3678 G-15
High affinity and selective GPER antagonist
4759 G-36
Selective GPER antagonist
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