p53 Activators

Cat. No. Product Name / Activity
3503 HLI 373
Hdm2 inhibitor; activates p53-dependent transcription
6904 Idasanutlin
Potent MDM2 inhibitor; inhibits MDM2-p53 interaction
6615 KCC 07
BAI1/p53 signaling activator; inhibits MBD2 (Methyl-CpG-binding domain protein 2)
5065 NSC 319726
Reactivator of mutant p53
3984 Nutlin-3
MDM2 antagonist; inhibits MDM2-p53 interaction
6075 Nutlin 3a
MDM2 antagonist; active enantiomer of Nutlin-3 (Cat. No. 3984)
2443 RITA
p53-MDM2 interaction inhibitor; antitumor
5332 SP 141
High affinity MDM2 inhibitor
3356 WR 1065 dihydrochloride
p53 activator. Also ROS scavenger