Cat. No. | Product Name / Activity |
---|---|
7256 | ARV 771 |
Potent BET bromodomain PROTAC®; also degrades BRD-tagged chimeric antigen receptors (CAR) in T cells | |
6356 | AT 1 |
(+)-JQ1 based PROTAC® with selectivity for BRD4 | |
7319 | BRD PHOTAC-I-3 |
Photoswitchable BET bromodomain degrader (PHOTAC) | |
7433 | cis-SIM1 |
Negative control for SIM1 (Cat. No. 7432) | |
6327 | dBET1 |
(+)-JQ1 based Degrader targeting BET bromodomains, active in vivo | |
6945 | dBET6 |
Potent and selective (+)-JQ1 based Degrader targeting BET bromodomains, active in vivo | |
6606 | dBRD9 |
Potent and selective BRD9 Degrader | |
6943 | dBRD9-A |
Potent BRD9 Degrader | |
6154 | MZ 1 |
BRD4 Degrader; preferentially degrades BRD4 over BRD2/3 | |
6936 | VZ 185 |
Potent and selective BRD7/9 Degrader |