Bromodomain Degraders

Cat. No. Product Name / Activity
7256 ARV 771
Potent BET bromodomain PROTAC®; also degrades BRD-tagged chimeric antigen receptors (CAR) in T cells
6356 AT 1
(+)-JQ1 based PROTAC® with selectivity for BRD4
7319 BRD PHOTAC-I-3
Photoswitchable BET bromodomain degrader (PHOTAC)
6327 dBET1
(+)-JQ1 based Degrader targeting BET bromodomains, active in vivo
6945 dBET6
Potent and selective (+)-JQ1 based Degrader targeting BET bromodomains, active in vivo
6606 dBRD9
Potent and selective BRD9 Degrader
6943 dBRD9-A
Potent BRD9 Degrader
7828 HHP 9
BET bromodomain degrader; also potent Hedgehog pathway inhibitor
6154 MZ 1
BRD4 Degrader; preferentially degrades BRD4 over BRD2/3
6936 VZ 185
Potent and selective BRD7/9 Degrader