Vasopressin Receptor Antagonists

Cat. No. Product Name / Activity
3377 (d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
Selective vasopressin V1A antagonist
6830 Conivaptan hydrochloride
Very high affinity vasopressin V1A and V2 antagonist; orally bioavailable
3924 OPC 21268
Orally active vasopressin V1 antagonist
2310 SR 49059
Selective, orally active vasopressin V1A receptor antagonist
6195 SSR 149415
Potent and selective vasopressin V1B antagonist
5729 TASP 0390325
Potent and selective V1B receptor antagonist; orally bioavailable
5181 Tolvaptan
Potent and selective vasopressin V2 receptor antagonist; renoprotective and orally active

Related Targets