GABA Inhibitors

Cat No Product Name / Activity
0206 β-Alanine
GABA uptake inhibitor (GAT-2 and -3). Also glycine receptor agonist
1296 CI 966 hydrochloride
Selective inhibitor of GAT-1
0234 Guvacine hydrochloride
Specific GABA uptake inhibitor
0236 (±)-Nipecotic acid
GABA uptake inhibitor
2747 NNC 05-2090 hydrochloride
GABA uptake inhibitor; moderately BGT-1 selective
1779 NNC 711
Selective GAT-1 inhibitor
0768 Riluzole hydrochloride
GABA uptake inhibitor; also inhibits glutamate release and blocks NaV channels
1081 SKF 89976A hydrochloride
Potent GAT-1 inhibitor; brain penetrant
1561 (S)-SNAP 5114
GABA uptake inhibitor
0181 TACA
GABA uptake inhibitor. Also GABAA agonist and substrate for GABA-T
4256 Tiagabine hydrochloride
Selective GAT-1 inhibitor; anticonvulsant