Cat. No. | Product Name / Activity |
---|---|
0206 | β-Alanine |
GABA uptake inhibitor (GAT-2 and -3); also glycine receptor agonist and MRGPRD agonist | |
1296 | CI 966 hydrochloride |
Selective inhibitor of GAT-1 | |
2747 | NNC 05-2090 hydrochloride |
GABA uptake inhibitor; moderately BGT-1 selective | |
1779 | NNC 711 |
Selective GAT-1 inhibitor | |
0768 | Riluzole hydrochloride |
GABA uptake inhibitor; also inhibits glutamate release and blocks NaV channels | |
1081 | SKF 89976A hydrochloride |
Potent GAT-1 inhibitor; brain penetrant | |
1561 | (S)-SNAP 5114 |
GABA uptake inhibitor | |
0181 | TACA |
GABA uptake inhibitor; also GABAA agonist and substrate for GABA-T | |
4256 | Tiagabine hydrochloride |
Selective GAT-1 inhibitor; anticonvulsant |