GABA Inhibitors
| Cat. No. | Product Name / Activity |
|---|---|
| 0206 | β-Alanine |
| GABA uptake inhibitor (GAT-2 and -3); also glycine receptor agonist and MRGPRD agonist | |
| 1296 | CI 966 hydrochloride |
| Selective inhibitor of GAT-1 | |
| 0234 | Guvacine hydrochloride |
| Specific GABA uptake inhibitor | |
| 2747 | NNC 05-2090 hydrochloride |
| GABA uptake inhibitor; moderately BGT-1 selective | |
| 1779 | NNC 711 |
| Selective GAT-1 inhibitor | |
| 0768 | Riluzole hydrochloride |
| GABA uptake inhibitor; also inhibits glutamate release and blocks NaV channels | |
| 1081 | SKF 89976A hydrochloride |
| Potent GAT-1 inhibitor; brain penetrant | |
| 1561 | (S)-SNAP 5114 |
| GABA uptake inhibitor | |
| 0181 | TACA |
| GABA uptake inhibitor; also GABAA agonist and substrate for GABA-T | |
| 4256 | Tiagabine hydrochloride |
| Selective GAT-1 inhibitor; anticonvulsant |
Pain Research Product Guide
Our Pain guide highlights over 280 products for Pain research.
Request copyDownload PDFGABA Scientific Review
Our GABA review gives an overview of the structure and function of the GABA receptors, as well as highlighting pharmacological ligands for their study.
Request copyDownload PDFAddiction Life Science Poster
Written by Prof David Nutt, this poster summarizes the brain circuits and neurotransmitter systems that are affected by the main classes of addictive drugs.
Request copyDownload PDFEpilepsy Life Science Poster
Written by Alsa Pitkänen and Xavier Ekolle Ndode-Ekane, this poster summarizes current knowledge about how epilepsy develops.
Request copyDownload PDFSchizophrenia Life Science Poster
Written by Justin M. Saunders and Javier González-Maeso
Our Schizophrenia poster highlights the targets and pathways representing the most promising strategies to pursue for novel drug development.
Request copyDownload PDF