GABA Inhibitors

Cat. No. Product Name / Activity
1296 CI 966 hydrochloride
Selective inhibitor of GAT-1
1779 NNC 711
Selective GAT-1 inhibitor
0768 Riluzole hydrochloride
GABA uptake inhibitor; also inhibits glutamate release and blocks NaV channels
1081 SKF 89976A hydrochloride
Potent GAT-1 inhibitor; brain penetrant
1561 (S)-SNAP 5114
GABA uptake inhibitor
0181 TACA
GABA uptake inhibitor; also GABAA agonist and substrate for GABA-T
4256 Tiagabine hydrochloride
Selective GAT-1 inhibitor; anticonvulsant