GABA Inhibitors
| Cat No | Product Name / Activity |
|---|---|
| 0206 | β-Alanine |
| GABA uptake inhibitor (GAT-2 and -3). Also glycine receptor agonist and MRGPRD agonist | |
| 1296 | CI 966 hydrochloride |
| Selective inhibitor of GAT-1 | |
| 0234 | Guvacine hydrochloride |
| Specific GABA uptake inhibitor | |
| 2747 | NNC 05-2090 hydrochloride |
| GABA uptake inhibitor; moderately BGT-1 selective | |
| 1779 | NNC 711 |
| Selective GAT-1 inhibitor | |
| 0768 | Riluzole hydrochloride |
| GABA uptake inhibitor; also inhibits glutamate release and blocks NaV channels | |
| 1081 | SKF 89976A hydrochloride |
| Potent GAT-1 inhibitor; brain penetrant | |
| 1561 | (S)-SNAP 5114 |
| GABA uptake inhibitor | |
| 0181 | TACA |
| GABA uptake inhibitor. Also GABAA agonist and substrate for GABA-T | |
| 4256 | Tiagabine hydrochloride |
| Selective GAT-1 inhibitor; anticonvulsant |
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