EZH2 Inhibitors

Cat. No. Product Name / Activity
4703 3-Deazaneplanocin A hydrochloride
EZH2 histone methyltransferase inhibitor
6790 GSK 126
Very high affinity and selective EZH2 inhibitor
6128 GSK 343
Potent and selective SAM-competitive EZH2 inhibitor
6153 JQEZ5
Potent and selective SAM-competitive EZH2 inhibitor
6169 PF 06726304 acetate
Highly potent and SAM-competitive EZH2 inhibitor
6708 SAH-EZH2
EZH2/EDD interaction inhibitor; suppresses PCR2 complex function
4904 UNC 1999
Potent and selective EZH2/EZH1 inhibitor
4930 UNC 2399
Biotinylated UNC 1999 (Cat.No. 4904)