Cyclin-Dependent Protein Kinase Inhibitors

Cat No Product Name / Activity
6400 Alsterpaullone
Potent cdk1 and cdk2 inhibitor; also inhibits GSK-3β and Lck
2072 Aminopurvalanol A
Selective cdk inhibitor; potently inhibits cdk1, cdk2 and cdk5
2457 Arcyriaflavin A
Potent cdk4 inhibitor; also potently inhibits CaM kinase II; antiviral
3968 AZD 5438
Cdk inhibitor; potently inhibits cdk1, 2, 5 and 9
3194 BIO
Cdk inhibitor; also potent GSK-3 inhibitor
5654 BMS 265246
Cdk inhibitor; potently inhibits cdk1 and cdk2
6438 BRD 6989
Cdk8 inhibitor; enhances IL-10 production
5608 BS 181 dihydrochloride
Selective cdk7 inhibitor
5471 CGP 60474
Potent cdk inhibitor
5472 CGP 74514 dihydrochloride
Potent cdk1 inhibitor
3605 (R)-CR8
Cdk inhibitor; potently inhibits cdk1 and cdk2; also inhibits CK1
6174 CVT 313
Cdk2 and cdk5 inhibitor
3610 (R)-DRF053 dihydrochloride
Cdk inhibitor; also potent CK1 inhibitor
3094 Flavopiridol hydrochloride
Cdk inhibitor; potently inhibits cdk2 and cdk9
1813 Indirubin-3'-oxime
Cdk inhibitor; also inhibits GSK-3β and other protein kinases
1398 Kenpaullone
Cdk inhibitor; also inhibits GSK-3β
6752 LDC 000067
Potent and selective CDK9 inhibitor
2152 NSC 625987
Cdk4 inhibitor
1867 NSC 663284
Cdc25 phosphatase inhibitor; blocks cdk1 and cdk2 activation
1937 NSC 693868
Cdk inhibitor; also inhibits GSK-3
3135 NU 2058
Cdk1 and cdk2 inhibitor
3301 NU 6140
Cdk2 inhibitor; also potent inhibitor of aurora kinase A and B
6535 NVP 2
Potent and selective ATP-competitive CDK9 inhibitor
1284 Olomoucine
Cdk inhibitor
1902 [Ala92]-p16 (84-103)
Cdk inhibitor
4786 PD 0332991 isethionate
Potent cdk4 and cdk6 inhibitor; brain penetrant
3140 PHA 767491 hydrochloride
Cdk inhibitor; potently inhibits cdk9; also inhibits MK2
1580 Purvalanol A
Cdk inhibitor; potently inhibits cdk1, cdk2 and cdk5
1581 Purvalanol B
Selective cdk inhibitor; potently inhibits cdk1, cdk2 and cdk5
5494 R 547
Potent and selective cdk inhibitor; orally bioavailable
4181 Ro 3306
Cdk1 inhibitor
1332 Roscovitine
Cdk inhibitor
2609 Ryuvidine
Cdk4 inhibitor; also SETD8 inhibitor
4875 Senexin A
Cdk8 inhibitor
4075 SNS 032
Cdk inhibitor; potently inhibits cdk2, cdk7 and cdk9
2907 SU 9516
Cdk inhibitor; potently inhibits cdk1 and cdk2