5-HT2C Receptor Antagonists

Cat No Product Name / Activity
0444 Clozapine
5-HT2A and 5-HT2C antagonist; also dopamine antagonist
1007 N-Desmethylclozapine
5-HT2C antagonist
1644 Mesulergine hydrochloride
5-HT2A and 5-HT2C antagonist; also dopamine receptor partial agonist
1050 RS 102221 hydrochloride
Selective 5-HT2C antagonist
1371 SB 200646 hydrochloride
5-HT2C/2B antagonist
1661 SB 206553 hydrochloride
Potent and selective 5-HT2B and 5-HT2C antagonist; orally active
1374 SB 215505
5-HT2B/2C antagonist
1379 SB 221284
Potent and selective 5-HT2B and 5-HT2C antagonist
1375 SB 228357
5-HT2C/2B antagonist/inverse agonist
2901 SB 242084
Selective 5-HT2C antagonist; brain penetrant
1255 SDZ SER 082 fumarate
Selective 5-HT2B/2C antagonist