Non-selective 5-HT2

Agonists

Cat No Product Name / Activity
2863 DOB hydrochloride
Selective 5-HT2 agonist
4797 Org 37684
5-HT2 agonist

Antagonists

Cat No Product Name / Activity
0524 AMI-193
Selective 5-HT2 antagonist
0460 Cinanserin hydrochloride
Selective 5-HT2 antagonist
0996 Cyproheptadine hydrochloride
5-HT2 antagonist
1523 LY 215840
5-HT2/5-HT7 antagonist
0590 Metergoline
5-HT2 antagonist. Also 5-HT1 antagonist and 5-HT1D ligand. Has moderate affinity for 5-HT6 and high affinity for 5-HT7
0997 Mianserin hydrochloride
5-HT2 antagonist. Has moderate affinity for 5-HT6
2018 Mirtazapine
Potent 5-HT2 antagonist. Also 5-HT3, H1 and α2-antagonist. Antidepressant
4349 Olanzapine
5-HT2A/D2 antagonist; atypical antipsychotic
4735 Quetiapine hemifumarate
5-HT2/D2 antagonist; atypical antipsychotic
1955 Ritanserin
Potent 5-HT2 antagonist