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SAG dihydrochloride

Cat. No. 6390 Submit a Review Datasheet / COA / SDS
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Cat.No. 6390 - SAG dihydrochloride | C28H28ClN3OS.2HCl
Description: Dihydrochloride salt of SAG; Smo receptor agonist
Chemical Name: 3-Chloro-N-[trans-4-(methylamino)cyclohexyl]-N-[[3-(4-pyridinyl)phenyl]methyl]benzo[b]thiophene-2-carboxamide dihydrochloride
Purity: ≥99% (HPLC)
Datasheet
Citations
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Literature
Biological Activity Technical Data Solubility Calculators Datasheets References

Biological Activity

Dihydrochloride salt of SAG; a potent Smoothened (Smo) receptor agonist.

Technical Data

M. Wt 562.98
Formula C28H28ClN3OS.2HCl
Storage Store at -20°C
Purity ≥99% (HPLC)
PubChem ID 71433770
InChI Key IYXUQUYRWPGIQL-UHFFFAOYSA-N
Smiles ClC1=C(C(N([C@H]2CC[C@H](NC)CC2)CC3=CC=CC(C4=CC=NC=C4)=C3)=O)SC5=CC=CC=C51

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 56.3 100
DMSO 56.3 100

Preparing Stock Solutions

The following data is based on the product molecular weight 562.98. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.78 mL 8.88 mL 17.76 mL
5 mM 0.36 mL 1.78 mL 3.55 mL
10 mM 0.18 mL 0.89 mL 1.78 mL
50 mM 0.04 mL 0.18 mL 0.36 mL

Molarity Calculator

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Product Datasheets

Certificate of Analysis / Product Datasheet
Safety Datasheet

References

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Citations for SAG dihydrochloride

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