N-Benzylnaltrindole hydrochloride

Discontinued Product

0754 has been discontinued.

Description: Selective non-peptide δ2 antagonist
Chemical Name: 1'-Benzyl-17-(cyclopropylmethyl)-6,7-didehydro-4,5a-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan hydrochloride
Datasheet
Citations
Reviews
Literature (2)

Biological Activity for N-Benzylnaltrindole hydrochloride

N-Benzylnaltrindole hydrochloride is a potent δ2-selective opioid receptor antagonist with a long duration of action in vivo.

Technical Data for N-Benzylnaltrindole hydrochloride

M. Wt 541.09
Formula C33H32N2O3.HCl
Storage Store at RT
CAS Number 1206487-81-1
PubChem ID 90479740
InChI Key KDEBSUYWJUBPCB-ZHYTUUPESA-N
Smiles O[C@@]24[C@]3([C@@H]8C(N6CC7=CC=CC=C7)=C(C5=C6C=CC=C5)C4)C1=C(O8)C(O)=CC=C1CC2N(CC9CC9)CC3.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for N-Benzylnaltrindole hydrochloride

References for N-Benzylnaltrindole hydrochloride

References are publications that support the biological activity of the product.

Korlipara et al (1994) N-Benzylnaltrindoles as long acting δ-opioid receptor antagonists. J.Med.Chem. 37 1882 PMID: 8021928

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Keywords: N-Benzylnaltrindole hydrochloride, N-Benzylnaltrindole hydrochloride supplier, δ2-opioid, delta2-opioid, selective, non-peptide, antagonists, DOP, Receptors, OP1, Delta, Opioid, 0754, Tocris Bioscience

Citations for N-Benzylnaltrindole hydrochloride

Citations are publications that use Tocris products.

Currently there are no citations for N-Benzylnaltrindole hydrochloride.

Reviews for N-Benzylnaltrindole hydrochloride

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!

*Please note that Tocris will only send literature to established scientific business / institute addresses.


Peptides Involved in Appetite Modulation Scientific Review

Peptides Involved in Appetite Modulation Scientific Review

Written by Sonia Tucci, Lynsay Kobelis and Tim Kirkham, this review provides a synopsis of the increasing number of peptides that have been implicated in appetite regulation and energy homeostasis; putative roles of the major peptides are outlined and compounds available from Tocris are listed.

Addiction Poster

Addiction Poster

The key feature of drug addiction is the inability to stop using a drug despite clear evidence of harm. This poster describes the brain circuits associated with addiction, and provides an overview of the main classes of addictive drugs and the neurotransmitter systems that they target.