N-Benzylnaltrindole hydrochloride

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Cat.No. 0754 - N-Benzylnaltrindole hydrochloride | C33H32N2O3.HCl | CAS No. 1206487-81-1
Description: Selective non-peptide δ2 antagonist
Chemical Name: 1'-Benzyl-17-(cyclopropylmethyl)-6,7-didehydro-4,5a-epoxy-3,14-dihydroxyindolo[2',3':6,7]morphinan hydrochloride

Biological Activity

Potent δ2-selective opioid receptor antagonist with a long duration of action in vivo.

Technical Data

M. Wt 541.09
Formula C33H32N2O3.HCl
Storage Store at RT
CAS Number 1206487-81-1
PubChem ID 90479740
Smiles O[C@@]24[C@]3([C@@H]8C(N6CC7=CC=CC=C7)=C(C5=C6C=CC=C5)C4)C1=C(O8)C(O)=CC=C1CC2N(CC9CC9)CC3.Cl

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

Solvent Max Conc. mg/mL Max Conc. mM
DMSO 54.11 100

Preparing Stock Solutions

The following data is based on the product molecular weight 541.09. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.85 mL 9.24 mL 18.48 mL
5 mM 0.37 mL 1.85 mL 3.7 mL
10 mM 0.18 mL 0.92 mL 1.85 mL
50 mM 0.04 mL 0.18 mL 0.37 mL

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Product Datasheets

Safety Datasheet


References are publications that support the products' biological activity.

Korlipara et al (1994) N-Benzylnaltrindoles as long acting δ-opioid receptor antagonists. J.Med.Chem. 37 1882 PMID: 8021928

If you know of a relevant reference for N-Benzylnaltrindole hydrochloride, please let us know.

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View all δ Opioid Receptor Antagonists

Keywords: N-Benzylnaltrindole hydrochloride, supplier, δ2-opioid, delta2-opioid, selective, non-peptide, antagonists, DOP, Receptors, OP1, Delta, Opioid, Receptors, Delta, Opioid, Receptors, Tocris Bioscience

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