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Submit ReviewISOX INACT
Description: Negative control for PF-CBP1
Chemical Name: 5-(Dimethyl-1,2-oxazol-4-yl)-2-[2-(4-methoxyphenyl)ethyl]--4,6-dimethyl-1-[2-(morpholin-4-yl)ethyl]-1H-1,3-benzodiazole
Purity: ≥98% (HPLC)
Biological Activity for ISOX INACT
ISOX INACT is a negative control for PF CBP1. Exhibits negligible activity at CBP and BRD4.
Active Analog also available.
Licensing Information
Sold for research purposes under agreement from Pfizer Inc.
Technical Data for ISOX INACT
| M. Wt | 488.62 |
| Formula | C29H36N4O3 |
| Storage | Store at +4°C |
| Purity | ≥98% (HPLC) |
| PubChem ID | 121237856 |
| InChI Key | FTOHXUPHICJSCR-UHFFFAOYSA-N |
| Smiles | CC(ON=C1C)=C1C2=C(C)C(N=C(CCC3=CC=C(OC)C=C3)N4CCN5CCOCC5)=C4C=C2C |
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
Tocris products are intended for laboratory research use only, unless stated otherwise.
Product Datasheets for ISOX INACT
References for ISOX INACT
References are publications that support the biological activity of the product.
Chekler et al (2015) Transcriptional profiling of a selective CREB binding protein bromodomain inhibitor highlights therapeutic opportunities. Chem.Biol. 22 1588 PMID: 26670081
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Keywords: ISOX INACT, ISOX INACT supplier, ISOXINACT, negative, control, PFCBP1, bromodomains, CBP, BRD4, Bromodomains, 5808, Tocris Bioscience
Citations for ISOX INACT
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