Discontinued ProductUnfortunately GBLD 345 (Cat. No. 0770) has been withdrawn from sale for commercial reasons.
A high affinity benzodiazepine agonist (IC50 against diazepam = 1 nM).
|Storage||Store at RT|
The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.
All Tocris products are intended for laboratory research use only.
Preparing Stock Solutions
The following data is based on the product molecular weight 375.43. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.
|Concentration / Solvent Volume / Mass||1 mg||5 mg||10 mg|
|1 mM||2.66 mL||13.32 mL||26.64 mL|
|5 mM||0.53 mL||2.66 mL||5.33 mL|
|10 mM||0.27 mL||1.33 mL||2.66 mL|
|50 mM||0.05 mL||0.27 mL||0.53 mL|
References are publications that support the products' biological activity.
Davies et al (1992) Substituted imidazo[1,2-b]pyridazines. New compounds with activity at central and peripheral benzodiazepine receptors. Biochem.Pharmacol. 44 1555 PMID: 1358075
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Keywords: GBLD 345, supplier, High, affinity, benzodiazepine, agonists, GABAA, Receptors, GBLD345, GABAA, Receptors, GABAA, Receptors, Tocris Bioscience
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