Fentanyl citrate

Discontinued Product

Fentanyl citrate (Cat. No. 3247) has been withdrawn from sale for commercial reasons.
Description: Potent and selective μ agonist
Alternative Names: Phentanyl citrate
Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate
Purity: ≥99% (HPLC)
Literature (2)

Biological Activity for Fentanyl citrate

Potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.

Technical Data for Fentanyl citrate

M. Wt 528.59
Formula C22H28N2O.C6H8O7
Storage Store at RT
Purity ≥99% (HPLC)
CAS Number 990-73-8
PubChem ID 13810
Smiles O=C(O)C(O)(CC(O)=O)CC(O)=O.O=C(CC)N(C3=CC=CC=C3)C1CCN(CCC2=CC=CC=C2)CC1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Product Datasheets for Fentanyl citrate

References for Fentanyl citrate

References are publications that support the biological activity of the product.

Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113 PMID: 7475964

Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233 PMID: 12738037

Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054 PMID: 14557380

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Citations for Fentanyl citrate

Citations are publications that use Tocris products.

Currently there are no citations for Fentanyl citrate.

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!

*Please note that Tocris will only send literature to established scientific business / institute addresses.

Peptides Involved in Appetite Modulation Scientific Review

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Written by Sonia Tucci, Lynsay Kobelis and Tim Kirkham, this review provides a synopsis of the increasing number of peptides that have been implicated in appetite regulation and energy homeostasis; putative roles of the major peptides are outlined and compounds available from Tocris are listed.

Addiction Poster

Addiction Poster

The key feature of drug addiction is the inability to stop using a drug despite clear evidence of harm. This poster describes the brain circuits associated with addiction, and provides an overview of the main classes of addictive drugs and the neurotransmitter systems that they target.