Fentanyl citrate

Discontinued Product

Fentanyl citrate (Cat. No. 3247) has been withdrawn from sale for commercial reasons.
Cat.No. 3247 - Fentanyl citrate | C22H28N2O.C6H8O7 | CAS No. 990-73-8
Description: Potent and selective μ agonist
Alternative Names: Phentanyl citrate
Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate
Purity: ≥99% (HPLC)
Datasheet
Citations
Reviews
Literature (5)

Biological Activity

Potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.

Technical Data

M. Wt 528.59
Formula C22H28N2O.C6H8O7
Storage Store at RT
Purity ≥99% (HPLC)
CAS Number 990-73-8
PubChem ID 13810
InChI Key IVLVTNPOHDFFCJ-UHFFFAOYSA-N
Smiles O=C(O)C(O)(CC(O)=O)CC(O)=O.O=C(CC)N(C3=CC=CC=C3)C1CCN(CCC2=CC=CC=C2)CC1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

References

References are publications that support the biological activity of the product.

Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113 PMID: 7475964

Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233 PMID: 12738037

Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054 PMID: 14557380

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Citations for Fentanyl citrate

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Currently there are no citations for Fentanyl citrate.

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