Fentanyl citrate

Pricing Availability Delivery Time Qty
Cat.No. 3247 - Fentanyl citrate | C22H28N2O.C6H8O7 | CAS No. 990-73-8
Description: Potent and selective μ agonist
Alternative Names: Phentanyl citrate
Chemical Name: N-Phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamide citrate
Purity: ≥99% (HPLC)
Datasheet
Citations
Literature

Biological Activity

Potent and selective μ-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for μ-, δ- and κ-opioid receptors respectively). Displays antinociceptive activity in vivo.

Technical Data

M. Wt 528.59
Formula C22H28N2O.C6H8O7
Storage Store at RT
Purity ≥99% (HPLC)
CAS Number 990-73-8
PubChem ID 13810
InChI Key IVLVTNPOHDFFCJ-UHFFFAOYSA-N
Smiles O=C(O)C(O)(CC(O)=O)CC(O)=O.O=C(CC)N(C3=CC=CC=C3)C1CCN(CCC2=CC=CC=C2)CC1

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Solubility Data

Solvent Max Conc. mg/mL Max Conc. mM
Solubility
water 21.14 40

Preparing Stock Solutions

The following data is based on the product molecular weight 528.59. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.89 mL 9.46 mL 18.92 mL
5 mM 0.38 mL 1.89 mL 3.78 mL
10 mM 0.19 mL 0.95 mL 1.89 mL
50 mM 0.04 mL 0.19 mL 0.38 mL

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Product Datasheets

Safety Datasheet

References

References are publications that support the products' biological activity.

Zernig et al (1995) Receptor reserve and affinity of mu-opioid agonists in mouse antinociception: correlation with receptor binding. Life Sci. 57 2113 PMID: 7475964

Liu et al (2003) Opioid activity of C8813, a novel and potent opioid analgesic. Life Sci. 73 233 PMID: 12738037

Stevenson et al (2003) Opioid interactions in rhesus monkeys: effects of δ + μ and δ + κ agonists on schedule-controlled responding and thermal nociception. J.Pharmacol.Exp.Ther. 307 1054 PMID: 14557380


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Citations for Fentanyl citrate

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