ent-LP 99

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Cat.No. 5497 - ent-LP 99 | C26H30ClN3O4S | CAS No. 1808948-28-8
Description: Negative Control for LP 99
Chemical Name: N-[(2S,3R)-2-(4-Chlorophenyl)-1-(1,2-dihydro-1,4-dimethyl-2-oxo-7-quinolinyl)-6-oxo-3-piperidinyl]-2-methyl-1-propanesulfonamide
Purity: ≥98% (HPLC)
Literature (5)

Biological Activity for ent-LP 99

ent-LP 99 is a negative Control for LP 99 (Cat.No. 5496).

Licensing Information

This probe is supplied in conjunction with the Structural Genomics Consortium. For further characterization details, please visit the ent-LP 99 probe summary on the SGC website.

Compound Libraries for ent-LP 99

ent-LP 99 is also offered as part of the Tocriscreen 2.0 Max. Find out more about compound libraries available from Tocris.

Technical Data for ent-LP 99

M. Wt 516.05
Formula C26H30ClN3O4S
Storage Store at -20°C
Purity ≥98% (HPLC)
CAS Number 1808948-28-8
Smiles CC(C(C=C1)=C(N2C)C=C1N3[C@@H](C4=CC=C(Cl)C=C4)[C@H](NS(=O)(CC(C)C)=O)CCC3=O)=CC2=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

Tocris products are intended for laboratory research use only, unless stated otherwise.

Solubility Data for ent-LP 99

Solvent Max Conc. mg/mL Max Conc. mM
DMSO 51.6 100
ethanol 51.6 100

Preparing Stock Solutions for ent-LP 99

The following data is based on the product molecular weight 516.05. Batch specific molecular weights may vary from batch to batch due to the degree of hydration, which will affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.94 mL 9.69 mL 19.38 mL
5 mM 0.39 mL 1.94 mL 3.88 mL
10 mM 0.19 mL 0.97 mL 1.94 mL
50 mM 0.04 mL 0.19 mL 0.39 mL

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References for ent-LP 99

References are publications that support the biological activity of the product.

Clark et al (2015) LP99: discovery and synthesis of the first selective BRD7/9 bromodomain inhibitor. Angew.Chem.Int.Ed.Engl. 54 6217 PMID: 25864491

If you know of a relevant reference for ent-LP 99, please let us know.

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Citations for ent-LP 99

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Literature in this Area

Tocris offers the following scientific literature in this area to showcase our products. We invite you to request* your copy today!

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