DSLET

Discontinued Product

Unfortunately DSLET (Cat. No. 1170) has been withdrawn from sale for commercial reasons.
Cat.No. 1170 - DSLET | Tyr-D-Ser-Gly-Phe-Leu-Thr | CAS No. 75644-90-5
Description: Selective δ agonist peptide
Alternative Names: [D-Ser2, Leu5, Thr6]-enkephalin
Datasheet
Citations
Literature

Biological Activity

δ Opioid receptor agonist.

Technical Data

M. Wt 686.9
Formula C33H46N6O10
Sequence YSGFLT

(Modifications: Ser-2 = D-Ser)

Storage Desiccate at -20°C
CAS Number 75644-90-5
Smiles [H]N[C@@H](CC1=CC=C(O)C=C1)C(=O)N[C@H](CO)C(=O)NCC(=O)N[C@@H](CC1=CC=CC=C1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H]([C@@H](C)O)C(O)=O

The technical data provided above is for guidance only. For batch specific data refer to the Certificate of Analysis.

All Tocris products are intended for laboratory research use only.

Preparing Stock Solutions

The following data is based on the product molecular weight 686.9. Batch specific molecular weights may vary from batch to batch due to solvent of hydration, which will affect the solvent volumes required to prepare stock solutions.

Select a batch to recalculate based on the batch molecular weight:
Concentration / Solvent Volume / Mass 1 mg 5 mg 10 mg
1 mM 1.46 mL 7.28 mL 14.56 mL
5 mM 0.29 mL 1.46 mL 2.91 mL
10 mM 0.15 mL 0.73 mL 1.46 mL
50 mM 0.03 mL 0.15 mL 0.29 mL

Molarity Calculator

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*When preparing stock solutions always use the batch-specific molecular weight of the product found on the vial label and SDS / CoA (available online).

Reconstitution Calculator

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Dilution Calculator

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Product Datasheets

Certificate of Analysis / Product Datasheet
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Safety Datasheet

References

References are publications that support the products' biological activity.

Hiller et al (1996) Autoradiographic comparison of [3H]DPDPE and [3H]DSLET binding: evidence for distinct δ1 and δ2 opioid receptor populations in rat brain. Brain Res. 719 85 PMID: 8782867

Yukhananov et al (1994) Opiate withdrawal intensity correlates with the presence of DSLET high-affinity binding. Pharmacol.Biochem.Behav. 49 1109 PMID: 7886084

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Keywords: DSLET, supplier, Selective, δ-opioid, delta-opioid, agonist, peptide, DOP, Receptors, OP1, [D-Ser2,, Leu5,, Thr6]-enkephalin, Delta, Opioid, Receptors, Tocris Bioscience

Citations for DSLET

Citations are publications that use Tocris products.

Currently there are no citations for DSLET.

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Reviews

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Literature in this Area

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Pathways for DSLET

Protocols

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