Voltage-gated Sodium (NaV) Channel Peptides

Activators

Cat. No. Product Name / Activity
5941 OD1
Potent hNav1.4, rNav1.6 and rNav1.7 channel activator

Blockers

Cat. No. Product Name / Activity
4804 APETx2
NaV1.8 and NaV1.2 blocker; also blocks ASIC3 channels
4913 Jingzhaotoxin III
Selective NaV1.5 channel blocker
4914 Phrixotoxin 3
Potent blocker of NaV1.2, NaV1.3 and NaV1.5 channels
4023 ProTx II
Selective NaV1.7 channel blocker